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Fluorescence-Coupled Ubiquitination Assay as a High-Throughput Screening Strategy for Novel Cereblon Degraders 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 10, 页码: 10111-10127
作者:  Deng, Yanan;  Yang, Shiling;  Xu, Hesong;  Ding, Xiyao;  Xu, Ying;  Ye, Zhengzheng;  Chen, Yan;  Zhang, Zemin;  Lin, Jin;  Xiong, Huan;  Zhang, Zizhong;  Yang, Kun;  Hu, Yiran;  Xu, Ke;  Luo, Cheng;  Chen, Shijie;  Lin, Hua;  Li, Zhihai
收藏  |  浏览/下载:7/0  |  提交时间:2025/06/23
A patent review of BRD4 inhibitors (2020-present) 期刊论文
EXPERT OPINION ON THERAPEUTIC PATENTS, 2025, 页码: 16
作者:  Chen, Yanfang;  Zhou, Huanmin;  Yu, Jiamin;  Gao, Jing;  Xue, Shengyu;  Ding, Hong;  Lin, Hua;  Luo, Cheng
收藏  |  浏览/下载:17/0  |  提交时间:2025/04/01
BET  BRD4  inhibitor  cancer treatment  selectivity  
Discovery of SET domain-binding primary alkylamine-tethered degraders for the simultaneous degradation of NSD2-long and RE-IIBP isoforms 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 283, 页码: 17
作者:  Hu, Linghao;  Xu, Hesong;  Xu, Ye;  Chen, Haowen;  Jiang, Hanrui;  Xu, Dounan;  Zhang, Huimin;  Luo, Cheng;  Chen, Shijie;  Wang, Mingliang
收藏  |  浏览/下载:38/0  |  提交时间:2025/04/01
NSD2  RE-IIBP  Targeted protein degradation  Multiple myeloma  
Identifying a non-conserved site for achieving allosteric covalent inhibition of CECR2 期刊论文
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 16
作者:  Tang, Cai-ling;  Li, Yuan-qing;  Du, Xi-kun;  Fang, Xiao-xia;  Guang, Yi-man;  Li, Pei-zhuo;  Chen, Shuang;  Xue, Sheng-yu;  Yu, Jia-min;  Liu, Xiao-yi;  Luo, Yi-pan;  Zhou, Lan-xin;  Luo, Cheng;  Xiong, Huan;  Liang, Zhong-jie;  Ding, Hong
收藏  |  浏览/下载:24/0  |  提交时间:2025/04/01
dynamics simulation  CECR2  covalent inhibitor  allosteric effect  
Inhibited peroxidase activity of peroxiredoxin 1 by palmitic acid exacerbates nonalcoholic steatohepatitis in male mice 期刊论文
NATURE COMMUNICATIONS, 2025, 卷号: 16, 期号: 1, 页码: 19
作者:  Yin, Wen;  Xu, Heng;  Bai, Zhonghao;  Wu, Yue;  Zhang, Yan;  Liu, Rui;  Wang, Zhangzhao;  Zhang, Bei;  Shen, Jing;  Zhang, Hao;  Chen, Xin;  Ma, Danting;  Shi, Xiaofeng;  Yan, Lihui;  Zhang, Chang;  Jiang, Hualiang;  Chen, Kaixian;  Guo, Dean;  Niu, Wenyan;  Yin, Huiyong;  Zhang, Weiping J.;  Luo, Cheng;  Xie, Xiangyang
收藏  |  浏览/下载:21/0  |  提交时间:2025/04/01
Defining ortholog-specific UHRF1 inhibition by STELLA for cancer therapy 期刊论文
NATURE COMMUNICATIONS, 2025, 卷号: 16, 期号: 1, 页码: 22
作者:  Bai, Wenjing;  Xu, Jinxin;  Gu, Wenbin;  Wang, Danyang;  Cui, Ying;  Rong, Weidong;  Du, Xiaoan;  Li, Xiaoxia;  Xia, Cuicui;  Gan, Qingqing;  He, Guantao;  Guo, Huahui;  Deng, Jinfeng;  Wu, Yuqiong;  Yen, Ray-Whay Chiu;  Yegnasubramanian, Srinivasan;  Rothbart, Scott B.;  Luo, Cheng;  Wu, Linping;  Liu, Jinsong;  Baylin, Stephen B.;  Kong, Xiangqian
收藏  |  浏览/下载:30/0  |  提交时间:2025/04/01
A peptide-centric local stability assay enables proteome-scale identification of the protein targets and binding regions of diverse ligands 期刊论文
NATURE METHODS, 2024, 页码: 17
作者:  Li, Kejia;  Chen, Shijie;  Wang, Keyun;  Wang, Yan;  Xue, Lianji;  Ye, Yuying;  Fang, Zheng;  Lyu, Jiawen;  Zhu, Haiyang;  Li, Yanan;  Yu, Ting;  Yang, Feng;  Zhang, Xiaolei;  Guo, Siqi;  Ruan, Chengfei;  Zhou, Jiahua;  Wang, Qi;  Dong, Mingming;  Luo, Cheng;  Ye, Mingliang
收藏  |  浏览/下载:160/0  |  提交时间:2025/01/14
YTHDF1 loss in dendritic cells potentiates radiation- induced antitumor immunity via STING-dependent I IFN 期刊论文
JOURNAL OF CLINICAL INVESTIGATION, 2024, 卷号: 134, 期号: 23, 页码: 14
作者:  Wen, Chuangyu;  Wang, Liangliang;  Piffko, Andras;  Chen, Dapeng;  Yu, Xianbin;  Zawieracz, Katarzyna;  Bugno, Jason;  Yang, Kaiting;  Naccasha, Emile Z.;  Ji, Fei;  Wang, Jiaai;  Huang, Xiaona;  Luo, Stephen Y.;  Tan, Lei;  Shen, Bin;  Luo, Cheng;  Mcnerney, Megan E.;  Chmura, Steven J.;  Arina, Ainhoa;  Pitroda, Sean;  He, Chuan;  Liang, Hua Laura;  Weichselbaum, Ralph R.
收藏  |  浏览/下载:25/0  |  提交时间:2025/04/01
Targeting 5-Hydroxytryptamine Receptor 1A in the Portal Vein to Decrease Portal Hypertension 期刊论文
GASTROENTEROLOGY, 2024, 卷号: 167, 期号: 5, 页码: 993-1007
作者:  Zhu, Chang-Peng;  Liu, Shu-Qing;  Wang, Ke-Qi;  Xiong, Hai-Lin;  Aristu-Zabalza, Peio;  Boyer-Diaz, Zoe;  Feng, Ji-Feng;  Song, Shao-Hua;  Luo, Cheng;  Chen, Wan-Sheng;  Zhang, Xin;  Dong, Wei-Hua;  Gracia-Sancho, Jordi;  Xie, Wei-Fen
收藏  |  浏览/下载:7/0  |  提交时间:2025/06/04
Portal Hypertension  Portal Vein Smooth Muscle Cells  5-Hydroxytryptamine  HTR1A  Alverine  
A Highly Atom-Efficient Prodrug Approach to Generate Synergy between H2S and Nonsteroidal Anti-inflammatory Drugs and Improve Safety 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 19, 页码: 17350-17362
作者:  Peng, Wen;  Qin, Lixiao;  Wang, Tianci;  Sun, Yangqian;  Li, Zhen;  Lefer, David J.;  Luo, Cheng;  Ye, Fei;  Wang, Binghe;  Guo, Weiwei;  Zheng, Yueqin
收藏  |  浏览/下载:46/0  |  提交时间:2024/11/05
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