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Targeted characterisation of bioactive prenylated flavonoids from Ficus carica L. fruits 期刊论文
FOOD CHEMISTRY, 2025, 卷号: 483, 页码: 11
作者:  Yuan, Yue;  Li, Zuopeng;  Aisa, Haji Akber
收藏  |  浏览/下载:3/0  |  提交时间:2025/06/23
Figs  Targeted isolation  Prenylated flavonoids  Antioxidant  Anti-inflammatory  Antitubercular  
Heterocycle-fused phenylcyclohexylamines as novel multi-target antagonists of N-methyl-D-aspartate (NMDA) receptor and monoamine transporter for treating depression 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 291, 页码: 20
作者:  Zheng, Fuqiang;  Hu, Zhengtao;  Chen, Hai;  Cheng, Jiaxin;  Hou, Qiongqiong;  Zheng, Jiefang;  Gong, Xudong;  Ji, Jing;  Zayniddin, Nuriddinov;  Abduahadi, Safomuddin;  Mamateli, Obul;  Wang, Guan;  Li, Pengcheng;  Hu, Tianwen;  Tian, Guanghui;  Xu, Zhijian;  Zhu, Weiliang;  Aisa, Haji Akber;  Shen, Jingshan;  He, Yang
收藏  |  浏览/下载:6/0  |  提交时间:2025/06/23
Heterocycle-fused phenylcyclohexylamines  Multi-target antagonists  NMDAR  Monoamine transporter  Antidepressants  
Direct Reductive N-alkylation of Amines with Carboxylic Esters 期刊论文
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2024, 页码: 7
作者:  Zhang, Yuxuan;  Bonku, Emmanuel Mintah;  Yang, Xingbang;  Zhu, Fuqiang;  Jiang, Xiangrui;  Abduahadi, Safomuddin;  Yang, Peng;  Aisa, Haji Akber;  Shen, Jingshan;  Qin, Hongjian
收藏  |  浏览/下载:36/0  |  提交时间:2025/01/14
Direct reductive N-alkylation of amine  One-pot reaction  Grignard reagent  Amidation of ester  Cariprazine  
Iron-Catalyzed Cross-Coupling Reactions of Alkyl Grignard Reagents with Alkenyl Carbonate 期刊论文
ADVANCED SYNTHESIS & CATALYSIS, 2024, 页码: 8
作者:  Qin, Hongjian;  Yang, Xingbang;  Mintah Bonku, Emmanuel;  Zhu, Fuqiang;  Abduahadi, Safomuddin;  Yang, Peng;  Shen, Jingshan;  Akber Aisa, Haji
收藏  |  浏览/下载:21/0  |  提交时间:2024/12/11
Iron catalysis  Alkylation of alkenyl carbonates  Grignard reagents  Cross-coupling reactions  C(sp2)-C(sp3) bonds formation  
Design, synthesis, and biological evaluation of novel 1-amido-2-one-4-thio-deoxypyranose as potential antitumor agents for multiple myeloma 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2024, 卷号: 111, 页码: 16
作者:  Li, Xiaomei;  Zhang, Hui;  Dong, Sanfeng;  Gao, Xuejie;  Sun, Haiguo;  Zhou, Zhaoyin;  Hu, Ke;  Guo, Shushan;  Zhang, Qikai;  Guo, Zhufeng;  Bunu, Samuel Jacob;  Zhu, Jianming;  Li, Bo;  Zhang, Yong;  Shen, Jingshan;  Aisa, Haji Akber;  Xu, Zhijian;  Cai, Haiyan;  Shi, Jumei;  Zhu, Weiliang
收藏  |  浏览/下载:39/0  |  提交时间:2024/09/26
Multiple myeloma  1-amido-2-one-4-thio-deoxypyranose  TRIP13 inhibitor  In vivo activity  
An Improved Iodine-Catalyzed Aromatization Reaction and Its Application in the Synthesis of a Key Intermediate of Cannabidiol 期刊论文
SYNLETT, 2024, 页码: 6
作者:  Abduahadi, Safomuddin;  Bonku, Emmanuel Mintah;  Qin, Hongjian;  Odilov, Abdullajon;  Zhu, Fuqiang;  Aisa, Haji Akber;  Shen, Jingshan
收藏  |  浏览/下载:53/0  |  提交时间:2024/05/22
methyl olivetolate  potassium persulfate  aromatization  oxidation  iodine-catalyst  cannabidiol  
Discovery of a CB2 and 5-HT1A receptor dual agonist for the treatment of depression and anxiety 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 20
作者:  Yang, Wenjiao;  Gong, Xudong;  Sun, Haiguo;  Wu, Chunhui;  Suo, Jin;  Ji, Jing;  Jiang, Xiangrui;  Shen, Jingshan;  He, Yang;  Aisa, Haji Akber
收藏  |  浏览/下载:70/0  |  提交时间:2024/03/06
CB2R agonist  5-HT1AR agonist  CB1R antagonist  Antidepressant  Anxiolytic  
Repurposing of Rutan showed effective treatment for COVID-19 disease 期刊论文
FRONTIERS IN MEDICINE, 2023, 卷号: 10, 页码: 13
作者:  Salikhov, Shavkat I.;  Abdurakhmonov, Ibrokhim Y.;  Oshchepkova, Yuliya I.;  Ziyavitdinov, Jamolitdin F.;  Berdiev, Nodir Sh.;  Aisa, Haji Akber;  Shen, Jingshan;  Xu, Yechun;  Xu, H. Eric;  Jiang, Xiangrui;  Zhang, Leike;  Vypova, Natalia L.;  Allaberganov, Dilshod Sh.;  Tagayalieva, Nigora A.;  Musabaev, Erkin I.;  Ibadova, Gulnara A.;  Rajabov, Ilxom B.;  Lokteva, Lyubov M.
收藏  |  浏览/下载:59/0  |  提交时间:2024/01/26
COVID-19  SARS-CoV-2  3CLpro  RdRp  Rhus coriaria  Rutan  clinical trial  
Toad venom bufadienolides and bufotoxins: An updated review 期刊论文
DRUG DEVELOPMENT RESEARCH, 2023, 页码: 24
作者:  Asrorov, Akmal M.;  Kayumov, Muzaffar;  Mukhamedov, Nurkhodja;  Yashinov, Ansor;  Mirakhmetova, Ziyoda;  Huang, Yongzhuo;  Yili, Abulimiti;  Aisa, Haji Akber;  Tashmukhamedov, Mugrajitdin;  Salikhov, Shavkat;  Mirzaakhmedov, Sharafitdin
收藏  |  浏览/下载:43/0  |  提交时间:2023/10/17
arenobufagin  bufadienolides  bufalin  bufotalin  cinobufagin  cinobufotalin  gamabufotalin  
Three new feruloyl glucuronopyranosyl glycerols from Eriocaulon buergerianum with their anti-fibrotic effects on hepatic stellate cells 期刊论文
NATURAL PRODUCT RESEARCH, 2023, 卷号: 37, 期号: 6, 页码: 956-966
作者:  Zhang, Yong;  Li, Hao;  Xu, Zhijian;  Shi, Yulong;  Li, Bo;  Li, Jia;  Aisa, Haji Akber;  Zang, Yi;  Zhu, Weiliang
收藏  |  浏览/下载:66/0  |  提交时间:2024/03/27
Eriocaulon buergerianum  Eriocaulaceae  feruloyl glucuronopyranosyl glycerols  TGF-beta 1 receptor  hepatic fibrosis  
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