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One stone two birds: Introducing piperazine into a series of nucleoside derivatives as potent and selective PRMT5 inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 281, 页码: 18
作者:  Li, Huaxuan;  Yang, Hong;  Liu, Li;  Zheng, Jiahong;  Shi, Qiongyu;  Li, Bang;  Wang, Xingcan;  Zhang, Ying;  Zhou, Ruilin;  Zhang, Jian;  Chen, Zhong-Zhu;  Wang, Chang-Yun;  Wang, Yuanxiang;  Huang, Xun;  Liu, Zhiqing
收藏  |  浏览/下载:49/0  |  提交时间:2024/12/11
Protein arginine methyltransferase 5  Nucleoside derivatives  Piperazine  Metabolic stability  Symmetric dimethylarginines  
Discovery of a New-Generation S-Adenosylmethionine-Noncompetitive Covalent Inhibitor Targeting the Lysine Methyltransferase Enhancer of Zeste Homologue 2 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 11, 页码: 7629-7644
作者:  Zhang, Yi;  Yang, Hong;  Li, Bingbing;  Li, Jiayi;  Li, Huaxuan;  Shi, Qiongyu;  Li, Bang;  Wang, Zekun;  Zheng, Jiahong;  Zhang, Ying;  Dong, Hui;  Huang, Xun;  Wang, Yuanxiang
收藏  |  浏览/下载:52/0  |  提交时间:2023/10/17
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