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BMAL1/PGC1a4-FNDC5/irisin axis impacts distinct outcomes of time-of-day resistance exercise 期刊论文
JOURNAL OF SPORT AND HEALTH SCIENCE, 2025, 卷号: 14, 页码: 23
作者:  Guo, Mingwei;  Shen, Fei;  Guo, Xiaozhen;  Zhang, Jun;  Ma, Ying;  Wu, Xia;  Zuo, Hui;  Yao, Jing;  Hu, Yepeng;  Wang, Dongmei;  Li, Yu;  Li, Jin;  Qiu, Jin;  Yu, Jian;  Meng, Meiyao;  Zheng, Ying;  Chen, Xin;  Gong, Mingkai;  Liu, Kailin;  Jin, Ling;  Ren, Xiangyu;  Zhang, Qiang;  Zhao, Yu;  Gu, Xuejiang;  Shen, Feixia;  Li, Dali;  Gao, Liangcai;  Liu, Chang;  Zhou, Fei;  Li, Mian;  Wang, Jiqiu;  Ding, Shuzhe;  Ma, Xinran;  Lu, Jian;  Xie, Cen;  Xiao, Junjie;  Xu, Lingyan
收藏  |  浏览/下载:40/0  |  提交时间:2025/04/01
Daily variance  Circadian  Muscle strength  Metabolic benefits  Resistance exercise  
Heterocycle-fused phenylcyclohexylamines as novel multi-target antagonists of N-methyl-D-aspartate (NMDA) receptor and monoamine transporter for treating depression 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 291, 页码: 20
作者:  Zheng, Fuqiang;  Hu, Zhengtao;  Chen, Hai;  Cheng, Jiaxin;  Hou, Qiongqiong;  Zheng, Jiefang;  Gong, Xudong;  Ji, Jing;  Zayniddin, Nuriddinov;  Abduahadi, Safomuddin;  Mamateli, Obul;  Wang, Guan;  Li, Pengcheng;  Hu, Tianwen;  Tian, Guanghui;  Xu, Zhijian;  Zhu, Weiliang;  Aisa, Haji Akber;  Shen, Jingshan;  He, Yang
收藏  |  浏览/下载:6/0  |  提交时间:2025/06/23
Heterocycle-fused phenylcyclohexylamines  Multi-target antagonists  NMDAR  Monoamine transporter  Antidepressants  
Discovery of multi-chitinase inhibitors cinnamyl thiazolidinone compounds as candidates for insect growth regulators via ligand-based optimization strategies 期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2025, 卷号: 306, 页码: 14
作者:  Jiang, Zhiyang;  Shi, Dongmei;  Fu, Haoyu;  Li, Yan;  Zou, Renxuan;  He, Ziqi;  Shi, Jie;  Shen, Lijuan;  Tang, Bin;  Xu, Zhijian;  Yang, Qing;  Duan, Hongxia
收藏  |  浏览/下载:9/0  |  提交时间:2025/05/27
Multi-chitinase inhibitor  Cinnamaldehyde compounds  Thiazolidinone compounds  Ligand-based optimization  Insect growth regulators (IGRs)  
Targeting Two Odorant-Binding Proteins in Acyrthosiphon pisum: Discovery of Novel Jasmone Derivatives as Aphid Repellents 期刊论文
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2025, 卷号: 73, 期号: 19, 页码: 11998-12013
作者:  Zhu, Ziwei;  Li, Huilin;  Zhu, Wenya;  Du, Shaoqing;  Yang, Zhaokai;  Ren, Jianing;  Xu, Zhijian;  Duan, Hongxia
收藏  |  浏览/下载:2/0  |  提交时间:2025/06/23
odorant-binding proteins  jasmone derivatives  rational design  aphid repellents  insect behaviorregulators  
Design and Development of a Novel Oral 4′-Fluorouridine Double Prodrug VV261 against SFTSV 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 9, 页码: 9811-9826
作者:  Cheng, Yong;  Zheng, Wei;  Dong, Xinru;  Sun, Tengxiao;  Xu, Mengwei;  Xiang, Li;  Li, Jian;  Wang, Huilong;  Jian, Xiaoqin;  Yu, Jingjin;  Li, Pengcheng;  Hu, Tianwen;  Tian, Guanghui;  Jiang, Xiangrui;  Zhang, Leike;  Aisa, Haji A.;  Xie, Yuanchao;  Xiao, Gengfu;  Shen, Jingshan
收藏  |  浏览/下载:1/0  |  提交时间:2025/06/23
Dynamically chiral phosphonic acid-type metallo-β-lactamase inhibitors 期刊论文
COMMUNICATIONS CHEMISTRY, 2025, 卷号: 8, 期号: 1, 页码: 13
作者:  Gulyas, Kinga Virag;  Zhou, Liping;  Salamonsen, Daniel;  Prester, Andreas;  Bartels, Kim;  Bosman, Robert;  Haffke, Paul;  Li, Jintian;  Tamasi, Viola;  Deufel, Fritz;  Thoma, Johannes;  Andersson Rasmussen, Anna;  Csala, Miklos;  Leiros, Hanna-Kirsti Schroder;  Xu, Zhijian;  Widersten, Mikael;  Rohde, Holger;  Schulz, Eike C.;  Zhu, Weiliang;  Erdelyi, Mate
收藏  |  浏览/下载:1/0  |  提交时间:2025/06/23
Discovery of 2,4-quinazolinedione derivatives as LC3B recruiters in the facilitation of protein complex degradations 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 287, 页码: 10
作者:  Zeng, Yanping;  Xiao, Jian;  Shi, Li;  Li, Yangsha;  Xu, Yuanxin;  Zhou, Jiayun;  Dong, Xiao;  Hou, Haiyang;  Zhong, Chao;  Cheng, Gang;  Chen, Yi;  Zhang, Naixia;  Fang, Yanfen;  Hu, Youhong
收藏  |  浏览/下载:21/0  |  提交时间:2025/04/01
LC3B  CDK9  Degradation  Protein complex  
Development of RelB-targeting small-molecule inhibitors of non-canonical NF-kB signaling with antitumor efficacy 期刊论文
MOLECULAR THERAPY, 2025, 卷号: 33, 期号: 4, 页码: 1519-1534
作者:  Li, Cuifeng;  Wei, Shuqi;  Sun, Donglin;  Yang, Zhuo;  Wang, Qi;  Lin, Han;  Zhang, Haohao;  Hu, Yiming;  Liu, Dandan;  Ye, Deji;  Tao, Yu;  Liu, Zhanjie;  Xu, Zhijian;  Li, Bo;  Li, Lingling;  Zhang, Jie;  Chen, Xi;  Xie, Ningxia;  Shi, Yufang;  Liu, Sanhong;  Liu, Yongzhong;  Jiang, Yuhang;  Zhu, Weiliang;  Zhang, Xiaoren
收藏  |  浏览/下载:18/0  |  提交时间:2025/05/27
Jatrophane and ingenane diterpenoids with anti-inflammatory activity from Euphorbia esula 期刊论文
PHYTOCHEMISTRY, 2025, 卷号: 232, 页码: 13
作者:  Li, Yu-Peng;  Li, Ying;  Gao, Wen-Jing;  Fang, Chu-Hong;  Lv, Ming-Jun;  Yue, Jian-Min;  Yu, Jin-Hai
收藏  |  浏览/下载:10/0  |  提交时间:2025/04/01
Euphorbia esula L.  Euphorbiaceae  Diterpenoid  Anti-inflammatory  NF-kappa B/MAPK  Nrf2/HO-1  
USP7 V517F mutation as a mechanism of inhibitor resistance 期刊论文
NATURE COMMUNICATIONS, 2025, 卷号: 16, 期号: 1, 页码: 14
作者:  Miao, Yu-Ling;  Fan, Fengying;  Cheng, Yong-Jun;  Jia, Li;  Song, Shan-Shan;  Huan, Xia-Juan;  Bao, Xu-Bin;  Ding, Jian;  Yu, Xuekui;  He, Jin-Xue
收藏  |  浏览/下载:8/0  |  提交时间:2025/05/27
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