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Dehydrotrametenolic acid methyl ester, a triterpenoid of Poria cocos, alleviates non-alcoholic steatohepatitis by suppressing NLRP3 inflammasome activation via targeting Caspase-1 in mice 期刊论文
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 17
作者:  Xia, Ling-yan;  Yu, Nai-rong;  Huang, Su-ling;  Qu, Hui;  Qin, Li;  Zhao, Qin-shi;  Leng, Ying
收藏  |  浏览/下载:3/0  |  提交时间:2025/06/23
non-alcoholic steatohepatitis  dehydrotrametenolic acid methyl ester  NLRP3 inflammasome  caspase-1  macrophage-hepatocyte/HSC crosstalk  
Discovery of multi-chitinase inhibitors cinnamyl thiazolidinone compounds as candidates for insect growth regulators via ligand-based optimization strategies 期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2025, 卷号: 306, 页码: 14
作者:  Jiang, Zhiyang;  Shi, Dongmei;  Fu, Haoyu;  Li, Yan;  Zou, Renxuan;  He, Ziqi;  Shi, Jie;  Shen, Lijuan;  Tang, Bin;  Xu, Zhijian;  Yang, Qing;  Duan, Hongxia
收藏  |  浏览/下载:10/0  |  提交时间:2025/05/27
Multi-chitinase inhibitor  Cinnamaldehyde compounds  Thiazolidinone compounds  Ligand-based optimization  Insect growth regulators (IGRs)  
Proteogenomic characterization of non-functional clinically relevant subgroups 期刊论文
CANCER CELL, 2025, 卷号: 43, 期号: 4, 页码: 36
作者:  Ji, Shunrong;  Cao, Lihua;  Gao, Jing;  Du, Yang;  Ye, Zeng;  Lou, Xin;  Liu, Fen;  Zhang, Yehan;  Xu, Junfeng;  Shi, Xiaohan;  Wang, Huan;  Li, Penghao;  Li, Yikai;  Chen, Hongxu;  Yang, Zhicheng;  Gao, Suizhi;  Zhang, Wuhu;  Huang, Dan;  Ni, Shujuan;  Wei, Miaoyan;  Wang, Fei;  Wang, Yan;  Ding, Tian;  Jing, Desheng;  Fan, Guixiong;  Gong, Zhiyun;  Lu, Renquan;  Qin, Yi;  Chen, Jie;  Xu, Xiaowu;  Wang, Pei;  Zhang, Bing;  Ding, Li;  Robles, Ana I.;  Rodriguez, Henry;  Chang, David K.;  Hruban, Ralph H.;  Gao, Dong;  Gao, Daming;  Jin, Gang;  Zhou, Hu;  Wu, Jianmin;  Yu, Xianjun
收藏  |  浏览/下载:3/0  |  提交时间:2025/06/23
Discovery of 2,4-quinazolinedione derivatives as LC3B recruiters in the facilitation of protein complex degradations 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 287, 页码: 10
作者:  Zeng, Yanping;  Xiao, Jian;  Shi, Li;  Li, Yangsha;  Xu, Yuanxin;  Zhou, Jiayun;  Dong, Xiao;  Hou, Haiyang;  Zhong, Chao;  Cheng, Gang;  Chen, Yi;  Zhang, Naixia;  Fang, Yanfen;  Hu, Youhong
收藏  |  浏览/下载:23/0  |  提交时间:2025/04/01
LC3B  CDK9  Degradation  Protein complex  
Development of RelB-targeting small-molecule inhibitors of non-canonical NF-kB signaling with antitumor efficacy 期刊论文
MOLECULAR THERAPY, 2025, 卷号: 33, 期号: 4, 页码: 1519-1534
作者:  Li, Cuifeng;  Wei, Shuqi;  Sun, Donglin;  Yang, Zhuo;  Wang, Qi;  Lin, Han;  Zhang, Haohao;  Hu, Yiming;  Liu, Dandan;  Ye, Deji;  Tao, Yu;  Liu, Zhanjie;  Xu, Zhijian;  Li, Bo;  Li, Lingling;  Zhang, Jie;  Chen, Xi;  Xie, Ningxia;  Shi, Yufang;  Liu, Sanhong;  Liu, Yongzhong;  Jiang, Yuhang;  Zhu, Weiliang;  Zhang, Xiaoren
收藏  |  浏览/下载:18/0  |  提交时间:2025/05/27
Molecular mechanism of the arrestin-biased agonism of neurotensin receptor 1 by an intracellular allosteric modulator 期刊论文
CELL RESEARCH, 2025, 卷号: 35, 期号: 4, 页码: 284-295
作者:  Sun, Demeng;  Li, Xiang;  Yuan, Qingning;  Wang, Yuanxia;  Shi, Pan;  Zhang, Huanhuan;  Wang, Tao;  Sun, Wenjing;  Ling, Shenglong;  Liu, Yuanchun;  Lai, Jinglin;  Xie, Wenqin;  Yin, Wanchao;  Liu, Lei;  Xu, H. Eric;  Tian, Changlin
收藏  |  浏览/下载:10/0  |  提交时间:2025/05/27
A positive-sense single-stranded RNA virus acquired a negative-sense open reading frame through recombination 期刊论文
PLOS PATHOGENS, 2025, 卷号: 21, 期号: 4, 页码: 16
作者:  Dong, Xuan;  Zhang, Fan;  Wang, Yiting;  Li, Cixiu;  Li, Xuan;  Zhou, Chengyan;  Wang, Guohao;  Tian, Zhongshuai;  Gao, Jing;  Zhou, Hu;  Sui, Liying;  Nauwynck, Hans;  Sorgeloos, Patrick;  Holmes, Edward C.;  Huang, Jie;  Shi, Weifeng
收藏  |  浏览/下载:9/0  |  提交时间:2025/05/27
A holistic strategy for the in-depth discrimination and authentication of 16 citrus herbs and associated commercial products based on machine learning techniques and non-targeted metabolomics 期刊论文
JOURNAL OF CHROMATOGRAPHY A, 2025, 卷号: 1745, 页码: 12
作者:  Huang, Yu-shi;  An, Ya-ling;  Zheng, Yue-yuan;  Zhao, Wen-jie;  Song, Chun-qian;  Zhang, Li-jie;  Chen, Jie-ting;  Tang, Zi-jun;  Feng, Lin;  Li, Zhen-wei;  Liu, Xiao-kang;  Zhang, Dai-di;  Guo, De-an
收藏  |  浏览/下载:10/0  |  提交时间:2025/04/01
Citrus herbs  Discrimination  LC-MS  Machine learning  Differential markers  
Time-Dependent Regulation of Sleep-Wakefulness and Electroencephalographic Characteristics by Spontaneous Running in Male Mice 期刊论文
JOURNAL OF SLEEP RESEARCH, 2025, 页码: 16
作者:  Zhou, Wufang;  Zhou, Jialin;  Lu, Qianyu;  Wang, Long;  Liang, Yutao;  Xing, Ye;  Zhang, Zheng;  Yang, Jinshan;  Zhao, Wenxue;  Li, Xin;  Shi, Guangsen
收藏  |  浏览/下载:9/0  |  提交时间:2025/05/27
delta power  spontaneous running  theta wave  voluntary exercise  
Oral FPR2/ALX modulators tune myeloid cell activity to ameliorate mucosal inflammation in inflammatory bowel disease 期刊论文
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 16
作者:  Yang, Wen-sheng;  Liu, Qing;  Li, Yang;  Li, Guan-yi;  Lin, Shi;  Li, Jie;  Li, Lin-yu;  Li, Yuan;  Ge, Xi-lin;  Wang, Xiao-zhen;  Wu, Wei;  Yan, Jun;  Wang, Guang-fei;  Zhou, Qing-tong;  Liu, Qiang;  Wang, Ming-Wei;  Li, Zhi-ping
收藏  |  浏览/下载:17/0  |  提交时间:2025/04/24
IBD  FPR2/ALX  Quin-C1  Quin-C7  neutrophils  macrophages  
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