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Synthesis and biological evaluation of multimodal monoaminergic arylpiperazine derivatives with potential antidepressant profile 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 275, 页码: 16
作者:  Zheng, Jiefang;  Zhou, Liping;  Gong, Xudong;  Yang, Feipu;  Cheng, Jiaxin;  Ma, Rui;  Wu, Chunhui;  Xu, Zhijian;  Zhu, Weiliang;  He, Yang;  Shen, Jingshan
收藏  |  浏览/下载:265/0  |  提交时间:2024/08/22
Triple reuptake inhibitors  5-HT 1A R agonists  Antidepressants  Multimodal serotonergic compounds  
The antidepressant-like effect and proposed mechanism of action of TPN672MA, a novel serotonin-dopamine receptor modulator for the treatment of schizophrenia 期刊论文
PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, 2024, 卷号: 242, 页码: 13
作者:  Cheng, Jiaxin;  Wu, Chunhui;  Wang, Yu;  Wang, Zhen;  He, Yang;  Shen, Jingshan
收藏  |  浏览/下载:57/0  |  提交时间:2024/08/22
TPN672MA  5-HT 1A receptor agonist  D 2 /D 3 receptor partial agonist  5-HT 2A receptor antagonist  Antidepressant-like  Mechanism  
Cannabidiol exhibits anxiolytic-like effects and antipsychotic-like effects in mice models 期刊论文
NEUROSCIENCE LETTERS, 2024, 卷号: 826, 页码: 8
作者:  Shu, Guangzhao;  He, Yang;  Suo, Jin;  Wu, Chunhui;  Gong, Xudong;  Xiang, Yangyang;  Yang, Wenjiao;  Cheng, Jiaxin;  Wang, Yu;  Chen, Weiming;  Shen, Jingshan
收藏  |  浏览/下载:41/0  |  提交时间:2024/06/27
Cannabidiol  Stress-induced hyperthermia  Phencyclidine-induced negative symptoms of  schizophrenia model  5-HT 1A receptor  
Discovery of a CB2 and 5-HT1A receptor dual agonist for the treatment of depression and anxiety 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 20
作者:  Yang, Wenjiao;  Gong, Xudong;  Sun, Haiguo;  Wu, Chunhui;  Suo, Jin;  Ji, Jing;  Jiang, Xiangrui;  Shen, Jingshan;  He, Yang;  Aisa, Haji Akber
收藏  |  浏览/下载:71/0  |  提交时间:2024/03/06
CB2R agonist  5-HT1AR agonist  CB1R antagonist  Antidepressant  Anxiolytic  
Preventive and therapeutic benefits of nelfinavir in rhesus macaques and human beings infected with SARS-CoV-2 期刊论文
Signal Transduction and Targeted Therapy, 2023, 卷号: 8, 期号: 5, 页码: 2384-2391
作者:  Xu, Zhijian;  Shi, Danrong;  Han, Jianbao;  Ling, Yun;  Jiang, Xiangrui;  Lu, Xiangyun;  Li, Chuan(1.3);  Gong, Likun;  Ge, Guangbo;  Zhang, Yani;  Zang, Yi;  Song, Tianzhang;  Feng, Xiaoli;  Tian, Renrong;  Ji, Jia;  Zhu, Miaojin;  Wu, Nanping;  Wu, Chunhui;  Wang, Zhen;  Xu, Yechun;  Peng, Cheng;  Zheng, Min;  Yang, Junling;  Du, Feifei(1.3);  Wu, Junliang;  Wang, Peipei;  Shen, Jingshan;  Zhang, Jianliang;  Zheng, Yongtang;  Yao, Hangping;  Zhu, Weiliang
收藏  |  浏览/下载:52/0  |  提交时间:2024/03/27
Disruption of C/EBP beta-Clec7a axis exacerbates neuroinflammatory injury via NLRP3 inflammasome-mediated pyroptosis in experimental neuropathic pain 期刊论文
JOURNAL OF TRANSLATIONAL MEDICINE, 2022, 卷号: 20, 期号: 1, 页码: 19
作者:  Wu, Dan;  Zhang, Yanqiong;  Zhao, Chunhui;  Li, Qiuyue;  Zhang, Junhong;  Han, Jiaxin;  Xu, Zhijian;  Li, Junfang;  Ma, Yan;  Wang, Ping;  Xu, Haiyu
收藏  |  浏览/下载:93/0  |  提交时间:2023/04/10
C/EBP beta-Clec7a axis  Neuroinflammation  Neuropathic Pain  NLRP3 Inflammasome-mediated Pyroptosis  
TPN171H alleviates pulmonary hypertension via inhibiting inflammation in hypoxia and monocrotaline-induced rats 期刊论文
VASCULAR PHARMACOLOGY, 2022, 卷号: 145, 页码: 11
作者:  Zhao, Congke;  Hu, Liqing;  He, Xiangrong;  Li, Lijun;  Yin, Minghui;  Tettey, Abraham Terkpertey;  Wang, Yu;  Shen, Jingshan;  Tang, Siyuan;  Wu, Chunhui;  Li, Qianbin;  Wang, Zhen;  Li, Xiaohui
收藏  |  浏览/下载:81/0  |  提交时间:2022/08/16
Pulmonary hypertension  Hypoxia  Monocrotaline  Anti-inflammatory effects  NLRP3 inflammasome  Pulmonary artery endothelial cells  
Disruption of C 期刊论文
JOURNAL OF TRANSLATIONAL MEDICINE, 2022, 卷号: 20, 期号: 1
作者:  Dan Wu;  Yanqiong Zhang;  Chunhui Zhao;  Qiuyue Li;  Junhong Zhang;  Jiaxin Han;  Zhijian Xu;  Junfang Li;  Yan Ma;  Ping Wang;  Haiyu Xu
收藏  |  浏览/下载:78/0  |  提交时间:2023/05/22
TPN672: A Novel Serotonin-Dopamine Receptor Modulator for the Treatment of Schizophrenia 期刊论文
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2021, 卷号: 378, 期号: 1, 页码: 20-30
作者:  Wang, Yu;  He, Yang;  Yang, Feipu;  Abame, Melkamu Alemu;  Wu, Chunhui;  Peng, Yanmin;  Feng, Linyin;  Shen, Jingshan;  Wang, Zhen;  He, Ling
收藏  |  浏览/下载:71/0  |  提交时间:2021/11/04
Chronic administration of synthetic cannabidiol induces antidepressant effects involving modulation of serotonin and noradrenaline levels in the hippocampus 期刊论文
NEUROSCIENCE LETTERS, 2021, 卷号: 744, 页码: 7
作者:  Abame, Melkamu Alemu;  He, Yang;  Wu, Song;  Xie, Zhifei;  Zhang, Jian;  Gong, Xudong;  Wu, Chunhui;  Shen, Jingshan
收藏  |  浏览/下载:85/0  |  提交时间:2021/05/24
Synthetic cannabidiol  Depression  Serotonin  Noradrenaline  Nuclear factor kappa B  
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