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Design, synthesis and evaluation of thieno[3,2-d]pyrimidine derivatives as novel potent CDK7 inhibitors 期刊论文
BIOORGANIC CHEMISTRY, 2024, 卷号: 148, 页码: 15
作者:  Zhang, Hongjin;  Lin, Guohao;  Jia, Suyun;  Wu, Jianbo;  Zhang, Ying;  Tao, Yanxin;  Huang, Weixue;  Song, Meiru;  Ding, Ke;  Ma, Dawei;  Fan, Mengyang
收藏  |  浏览/下载:36/0  |  提交时间:2024/09/26
Cyclin-dependent kinase 7  Small molecular inhibitor  Triple negative breast cancer  Thieno[3,2-d]pyrimidine derivative  
Discovery and optimization of thieno[3,2-d]pyrimidine derivatives as highly selective inhibitors of cyclin-dependent kinase 7 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 263, 页码: 21
作者:  Zhang, Hongjin;  Lin, Guohao;  Jia, Suyun;  Zhang, Ying;  Wu, Jianbo;  Tao, Yanxin;  Huang, Weixue;  Song, Meiru;  Ding, Ke;  Ma, Dawei;  Fan, Mengyang
收藏  |  浏览/下载:61/0  |  提交时间:2024/01/26
Thieno[3  d ]pyrimidine derivative  Cyclin-dependent kinase 7  Small molecule inhibitor  Kinome selectivity  Triple negative breast cancer  
Effect of an Herbal-Based Injection on 28-Day Mortality in Patients With Sepsis The EXIT-SEP Randomized Clinical Trial 期刊论文
JAMA INTERNAL MEDICINE, 2023, 卷号: 183, 期号: 7, 页码: 647-655
作者:  Liu, Songqiao;  Yao, Chen;  Xie, Jianfeng;  Liu, Hong;  Wang, Hongliang;  Lin, Zhaofen;  Qin, Bingyu;  Wang, Difen;  Lu, Weihua;  Ma, Xiaochun;  Liu, Yan;  Liu, Ling;  Zhang, Chi;  Xu, Lei;  Zheng, Ruiqiang;  Zhou, Feihu;  Liu, Zhongmin;  Zhang, Guoqiang;  Zhou, Lixin;  Liu, Jian;  Fei, Aihua;  Zhang, Guoxiu;  Zhu, Yimin;  Qian, Kejian;  Wang, Ruilan;  Liang, Yafeng;  Duan, Meili;  Wu, Dawei;  Sun, Rongqing;  Wang, Ying;  Zhang, Xijing;  Cao, Quan;  Yang, Mingshi;  Jin, Minggen;  Song, Yan;  Huang, Ling;  Zhou, Fachun;  Chen, Dechang;  Liang, Qun;  Qian, Chuanyun;  Tang, Zhongzhi;  Zhang, Zhong;  Feng, Qiming;  Peng, Zhiyong;  Sun, Renhua;  Song, Zhenju;  Sun, Yunbo;  Chai, Yanfen;  Zhou, Lihua;  Cheng, Chen;  Li, Li;  Yan, Xiaoyan;  Zhang, Junhua;  Huang, Yingzi;  Guo, Fengmei;  Li, Chuan;  Yang, Yi;  Shang, Hongcai;  Qiu, Haibo;  EXIT-SEP Investigators
收藏  |  浏览/下载:58/0  |  提交时间:2024/03/27
Cyclobutane Derivatives As Novel Nonpeptidic Small Molecule Agonists of Glucagon-Like Peptide-1 Receptor 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2012, 卷号: 55, 期号: 1, 页码: 250-267
作者:  Liu, Qing;  Li, Na;  Yuan, Yunyun;  Lu, Huili;  Wu, Xiaoyan;  Zhou, Caihong;  He, Min;  Su, Haoran;  Zhang, Meng;  Wang, Jia;  Wang, Bao;  Wang, You;  Ma, Dawei;  Ye, Yang;  Weiss, Hans-Christoph;  Gesing, Ernst R. F.;  Liao, Jiayu;  Wang, Ming-Wei
收藏  |  浏览/下载:50/0  |  提交时间:2019/01/08
acontinuedsagaofboc5thefirstnonpeptidicglucagonlikepeptide1receptoragonistwithinvivoactivities 期刊论文
actapharmacologicasinica, 2012, 卷号: 33, 期号: 2, 页码: 148
作者:  He Min;  Guan Ni;  Gao Weiwei;  Liu Qing;  Wu Xiaoyan;  Ma Dawei;  Zhong Dafang;  Ge Guangbo;  Li Chuan;  Chen Xiaoyan;  Yang Ling;  Liao Jiayu;  Wang Mingwei
收藏  |  浏览/下载:57/0  |  提交时间:2020/07/01
Type 2 diabetes  Glucagon-like peptide-1  Non-peptidic agonist  Boc5  G-protein coupled receptor  
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