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Identification of CDKN1A as a potential key risk factor in MASLD progression 期刊论文
FASEB JOURNAL, 2025, 卷号: 39, 期号: 7, 页码: 15
作者:  Deng, Lijuan;  Deng, Jianxin;  Luo, Liping;  Yang, Hongjia;  Sun, Mengxue;  Gao, Yucheng;  Liu, Qing;  Ngowi, Ebenezeri Erasto;  Zhou, Yinghua;  Zhang, Rongrong;  Liu, Xiaojun;  Qiao, Aijun
收藏  |  浏览/下载:14/0  |  提交时间:2025/05/27
biomarkers  CDKN1A  liver  MASLD  RNA-seq  
Discovery of a potential hematologic malignancies therapy: Selective and potent HDAC7 PROTAC degrader targeting non-enzymatic function 期刊论文
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 3, 页码: 1659-1679
作者:  Jin, Yuheng;  Qi, Xuxin;  Yu, Xiaoli;  Cheng, Xirui;  Chen, Boya;  Wu, Mingfei;  Zhang, Jingyu;  Yin, Hao;  Lu, Yang;  Zhou, Yihui;  Pang, Ao;  Lin, Yushen;  Jiang, Li;  Shi, Qiuqiu;  Geng, Shuangshuang;  Zhou, Yubo;  Yao, Xiaojun;  Li, Linjie;  Duan, Haiting;  Che, Jinxin;  Cao, Ji;  He, Qiaojun;  Dong, Xiaowu
收藏  |  浏览/下载:2/0  |  提交时间:2025/06/23
HDAC7  PROTAC  Selectivity  Hematologic malignancies  Non-enzymatic function  
Ligand-Enabled Pd-Catalyzed sp3 C-H Macrocyclization: Synthesis and Evaluation of Macrocyclic Sulfonamide for the Treatment of Parkinson's Disease 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2024, 卷号: 63, 期号: 45, 页码: 11
作者:  Bi, Tongyu;  Cui, Yunxia;  Liu, Shuai;  Yu, Haiyue;  Qiu, Weirong;  Hou, Ke-Qiang;  Zou, Jiaqi;  Yu, Zhipeng;  Zhang, Feili;  Xu, Zhongliang;  Zhang, Jian;  Xu, Xiaojun;  Yang, Weibo
收藏  |  浏览/下载:49/0  |  提交时间:2024/11/26
C-H activation  ligand-mediated macrocyclization  Pd catalysis  SIRT3  PD treatment  
LncRNA-Snhg3 regulates mouse hepatic glycogenesis under normal chow diet 期刊论文
FASEB JOURNAL, 2024, 卷号: 38, 期号: 15, 页码: 15
作者:  Xie, Xianghong;  Gao, Mingyue;  Wang, Heping;  Zhang, Minglong;  Zhao, Wei;  Li, Chunmei;  Zhang, Weihong;  Yang, Jiahui;  Zhang, Yinliang;  Chen, Enhui;  Guo, Yanfang;  Guo, Zeyu;  Ngowi, Ebenezeri Erasto;  Wang, Xiaoman;  Zhu, Yinghan;  Wang, Yiting;  Li, Xiaolu;  Yao, Hong;  Yan, Li;  Fang, Fude;  Li, Meixia;  Qiao, Aijun;  Liu, Xiaojun
收藏  |  浏览/下载:48/0  |  提交时间:2024/09/26
chromatin remodeling  glycogenesis  insulin resistance  lncRNA-Snhg3  
Discovery of a Highly Potent and Selective BRD9 PROTAC Degrader Based on E3 Binder Investigation for the Treatment of Hematological Tumors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 28
作者:  Duan, Haiting;  Zhang, Jingyu;  Gui, Renzhao;  Lu, Yang;  Pang, Ao;  Chen, Beijing;  Shen, Liteng;  Yu, Hengyuan;  Li, Jia;  Xu, Tengfei;  Wang, Yuwei;  Yao, Xiaojun;  Zhang, Bo;  Lin, Nengming;  Dong, Xiaowu;  Zhou, Yubo;  Che, Jinxin
收藏  |  浏览/下载:62/0  |  提交时间:2024/08/20
Qing-Zhi-Tiao-Gan-Tang (QZTGT) prevents nonalcoholic steatohepatitis (NASH) by expression pattern correction 期刊论文
JOURNAL OF ETHNOPHARMACOLOGY, 2023, 卷号: 317, 页码: 14
作者:  Chu, Hang;  Zhang, Weitao;  Tan, Yan;  Diao, Zhipeng;  Li, Peng;  Wu, Yapeng;  Xie, Like;  Sun, Jianguo;  Yang, Ke;  Li, Pingping;  Xie, Cen;  Li, Ping;  Hua, Qian;  Xu, Xiaojun
收藏  |  浏览/下载:86/0  |  提交时间:2023/10/17
Fibrosis  Inflammation  Lipogenesis  NASH  QZTGT  TMNP  
Saikosaponin D improves nonalcoholic fatty liver disease via gut microbiota-bile acid metabolism pathway 期刊论文
Food Science and Human Wellness, 2023
作者:  Li, Lan;  Yang, Shengye;  Liang, Xinyu;  Liu, Yameng;  Xu, Hualing;  Guo, Xiaozhen;  Xie, Cen;  Xu, Xiaojun
收藏  |  浏览/下载:96/0  |  提交时间:2024/03/26
Gut Microbiota  Non-alcoholic Fatty Liver Disease  Ssd  Bile Acids  Farnesoid x Receptor  
Trifluoroacetic Anhydride as Acylating Agent and Dehydrant in One-pot Synthesis of Nirmatrelvir 期刊论文
INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY, 2022, 卷号: 32, 期号: 4, 页码: 429-432
作者:  Jin, Chen;  Zhaug, Yan;  Li, Rui;  Yang, Xiaojun;  Zhu, Fuqiang;  Jiang, Xiangrui;  Zhang, Qiumeng;  Shen, Jingshan
收藏  |  浏览/下载:71/0  |  提交时间:2023/04/10
Discovery of a novel protein kinase C activator from Croton tiglium for inhibition of non-small cell lung cancer 期刊论文
PHYTOMEDICINE, 2019, 卷号: 65, 页码: 11
作者:  Wang Yuwei;  Tang Chunping;  Yao Sheng;  Lai Huanling;  Li Runze;  Xu Jiahui;  Wang Qianqian;  Fan Xing Xing;  Wu Qi Biao;  Lai-Han, Leung Elaine;  Ye Yang;  Yao Xiaojun
收藏  |  浏览/下载:87/0  |  提交时间:2020/07/01
Non-small cell lung cancer  Natural product  Croton tiglium  Protein kinase C  Molecular modelling  
Pharmacokinetics-Driven Optimization of 4(3H)-Pyrimidinones as Phosphodiesterase Type 5 Inhibitors Leading to TPN171, a Clinical Candidate for the Treatment of Pulmonary Arterial Hypertension 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 10, 页码: 4979-4990
作者:  Wang, Zhen;  Jiang, Xiangrui;  Zhang, Xianglei;  Tian, Guanghui;  Yang, Rulei;  Wu, Jianzhong;  Zou, Xiaoli;  Liu, Zheng;  Yang, Xiaojun;  Wu, Chunhui;  Shi, Jing;  Li, Jianfeng;  Suo, Jin;  Wang, Yu;  Zhang, Rongxia;  Xu, Zhijian;  Gong, Xudong;  He, Yang;  Zhu, Weiliang;  Aisa, Haji Akber;  Jiang, Hualiang;  Xu, Yechun;  Shen, Jingshan
收藏  |  浏览/下载:73/0  |  提交时间:2020/07/01
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