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中国科学院上海药物研究所机构知识库
Knowledge Management System of Shanghai Institute of Materia Medica, CAS
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Phytochemical and biological studies on rare and endangered plants endemic to China. Part XLIV. Integrated NMR/EI-MS/LC-PDA-ESIMS approach for dereplication and targeted isolation of fortunefuroic acids from
Keteleeria
fortunei
across diverse geographical origins
期刊论文
PHYTOCHEMISTRY, 2025, 卷号: 235, 页码: 13
作者:
Zhao, Ze-Yu
;
Jiang, Zhe-Lu
;
Tong, Ying-Peng
;
Chi, Chun-Jing
;
Zang, Yi
;
Choo, Yeun-Mun
;
Xiong, Juan
;
Li, Jia
;
Hu, Jin-Feng
收藏
|
浏览/下载:25/0
|
提交时间:2025/04/24
Keteleeria fortunei
Pinaceae
Geographical origins
Integrated NMR/EI-MS/LC-PDA-ESIMS
methods
Fortunefuroic acids
ATP-Citrate lyase
Pharmacokinetics and Safety of TPN171 (a PDE5 Inhibitor) in Patients With Mild or Moderate Hepatic Impairment Versus Participants With Normal Hepatic Function: A Phase I Study
期刊论文
CLINICAL PHARMACOLOGY IN DRUG DEVELOPMENT, 2025, 页码: 7
作者:
Zhou, Jing
;
Zhang, Hong
;
Ding, Yanhua
;
Wang, Zhen
;
Wang, Yu
;
Juan, Jiaxiang
;
Jiang, Zhicheng
;
Chen, Hong
收藏
|
浏览/下载:1/0
|
提交时间:2025/06/23
hepatic impairment
pharmacokinetics
phosphodiesterase-5 inhibitor
TPN171
A Phase I Study to Evaluate the Pharmacokinetics and Safety of TPN171 (a PDE5 Inhibitor) in Adults with Renal Impairment
期刊论文
CLINICAL PHARMACOLOGY IN DRUG DEVELOPMENT, 2025, 页码: 8
作者:
Fu, Ping
;
Song, Yi
;
Hu, Chao
;
Yong, Xiaolan
;
Yu, Yang
;
Chen, Yi
;
Wang, Ying
;
Zhu, Xiaohong
;
Wang, Zhen
;
Wang, Yu
;
Juan, Jiaxiang
;
Chen, Yuan
;
Miao, Jia
收藏
|
浏览/下载:2/0
|
提交时间:2025/06/23
pharmacokinetics
phosphodiesterase 5 inhibitor
renal impairment
safety
TPN171
USP7 V517F mutation as a mechanism of inhibitor resistance
期刊论文
NATURE COMMUNICATIONS, 2025, 卷号: 16, 期号: 1, 页码: 14
作者:
Miao, Yu-Ling
;
Fan, Fengying
;
Cheng, Yong-Jun
;
Jia, Li
;
Song, Shan-Shan
;
Huan, Xia-Juan
;
Bao, Xu-Bin
;
Ding, Jian
;
Yu, Xuekui
;
He, Jin-Xue
收藏
|
浏览/下载:9/0
|
提交时间:2025/05/27
New Arylalkenyl α-Pyrones from
Cryptocarya densiflora
期刊论文
CHEMISTRY & BIODIVERSITY, 2025, 页码: 6
作者:
Meng, Jie
;
Xue, Jun-Juan
;
Miao, Lei
;
Zhang, Yu
;
Rao, Li
;
Zhang, Chuan-Rui
收藏
|
浏览/下载:11/0
|
提交时间:2025/04/01
alpha-pyrones
Cryptocarya densiflora
cytotoxicity
quantum chemical calculations
spectroscopic data
Benzofurans and dibenzofurans from galls on twigs of the endangered Chinese endemic tree
Parrotia
subaequalis
and their inhibitory properties against
Staphylococcus
aureus
and ATP-citrate lyase
期刊论文
PHYTOCHEMISTRY, 2025, 卷号: 229, 页码: 9
作者:
Zhou, Peng-Jun
;
Wu, Xi-Ying
;
Zhao, Ze-Yu
;
Zang, Yi
;
Sun, Zhong-Shuai
;
Li, Yue-Ling
;
Li, Na
;
Xiong, Juan
;
Choo, Yeun-Mun
;
Jin, Ze-Xin
;
Li, Jia
;
Hu, Jin-Feng
收藏
|
浏览/下载:52/0
|
提交时间:2024/11/26
Parrotia subaequalis
Hamamelidaceae
Gall
Phytoalexins
Benzofuran
Dibenzofuran
Staphylococcus aureus
ATP-Citrate lyase
π-HuB: the proteomic navigator of the human body
期刊论文
NATURE, 2024, 卷号: 636, 期号: 8042, 页码: 322-331
作者:
He, Fuchu
;
Aebersold, Ruedi
;
Baker, Mark S.
;
Bian, Xiuwu
;
Bo, Xiaochen
;
Chan, Daniel W.
;
Chang, Cheng
;
Chen, Luonan
;
Chen, Xiangmei
;
Chen, Yu-Ju
;
Cheng, Heping
;
Collins, Ben C.
;
Corrales, Fernando
;
Cox, Juergen
;
Weinan, E.
;
Van Eyk, Jennifer E.
;
Fan, Jia
;
Faridi, Pouya
;
Figeys, Daniel
;
Gao, George Fu
;
Gao, Wen
;
Gao, Zu-Hua
;
Goda, Keisuke
;
Goh, Wilson Wen Bin
;
Gu, Dongfeng
;
Guo, Changjiang
;
Guo, Tiannan
;
He, Yuezhong
;
Heck, Albert J. R.
;
Hermjakob, Henning
;
Hunter, Tony
;
Iyer, Narayanan Gopalakrishna
;
Jiang, Ying
;
Jimenez, Connie R.
;
Joshi, Lokesh
;
Kelleher, Neil L.
;
Li, Ming
;
Li, Yang
;
Lin, Qingsong
;
Liu, Cui Hua
;
Liu, Fan
;
Liu, Guang-Hui
;
Liu, Yansheng
;
Liu, Zhihua
;
Low, Teck Yew
;
Lu, Ben
;
Mann, Matthias
;
Meng, Anming
;
Moritz, Robert L.
;
Nice, Edouard
;
Ning, Guang
;
Omenn, Gilbert S.
;
Overall, Christopher M.
;
Palmisano, Giuseppe
;
Peng, Yaojin
;
Pineau, Charles
;
Poon, Terence Chuen Wai
;
Purcell, Anthony W.
;
Qiao, Jie
;
Reddel, Roger R.
;
Robinson, Phillip J.
;
Roncada, Paola
;
Sander, Chris
;
Sha, Jiahao
;
Song, Erwei
;
Srivastava, Sanjeeva
;
Sun, Aihua
;
Sze, Siu Kwan
;
Tang, Chao
;
Tang, Liujun
;
Tian, Ruijun
;
Vizcaino, Juan Antonio
;
Wang, Chanjuan
;
Wang, Chen
;
Wang, Xiaowen
;
Wang, Xinxing
;
Wang, Yan
;
Weiss, Tobias
;
Wilhelm, Mathias
;
Winkler, Robert
;
Wollscheid, Bernd
;
Wong, Limsoon
;
Xie, Linhai
;
Xie, Wei
;
Xu, Tao
;
Xu, Tianhao
;
Yan, Liying
;
Yang, Jing
;
Yang, Xiao
;
Yates, John
;
Yun, Tao
;
Zhai, Qiwei
;
Zhang, Bing
;
Zhang, Hui
;
Zhang, Lihua
;
Zhang, Lingqiang
;
Zhang, Pingwen
;
Zhang, Yukui
;
Zheng, Yu Zi
;
Zhong, Qing
;
Zhu, Yunping
;
Tan, Chris Soon Heng
;
Gao, Mingxia
;
Gao, Qiang
;
Gao, Yushun
;
Guo, Xuejiang
;
He, Jie
;
He, Jun
;
He, Qing-Yu
;
Hou, Jinlin
;
Huang, Canhua
;
Jia, Chenxi
;
Kuster, Bernhard
;
Li, Chaoying
;
Li, Dong
;
Li, Yanchang
;
Liu, Siqi
;
Liu, Xiaonan
;
Liu, Ya
;
Liu, Zhongyang
;
Lu, Haojie
;
Nie, Yongzhan
;
Okada, Mariko
;
Qian, Guojun
;
Qin, Hongqiang
;
Rao, Yu
;
Rao, Zihe
;
Ren, Xianwen
;
Ren, Yan
;
Shen, Feng
;
Shen, Lin
;
Su, Shicheng
;
Tan, Minjia
;
Tang, Ben Zhong
;
Tao, Sheng-Ce
;
Wang, Jian
;
Wang, Tong
;
Wei, Liming
;
Wong, Catherine C. L.
;
Xie, Xiaoliang Sunney
;
Xu, Li
;
Xu, Ping
;
Yang, Huanming
;
Yang, Jianjun
;
Ye, Mingliang
;
Ying, Wantao
;
Yu, Xiaobo
;
Yuan, Yaxiang
;
Zeng, Qingcun
;
Zhan, Qimin
;
Zhang, Xiaofei
;
Zhang, Xu
;
Zhang, Ying
;
Zhong, Nan-Shan
;
Zhou, Feng
;
Zhu, Yi
;
Zhang, Zemin
收藏
|
浏览/下载:16/0
|
提交时间:2025/04/01
Optimization and Biological Evaluation of Novel 1
H
-Pyrrolo[2,3-
c
]pyridin Derivatives as Potent and Reversible Lysine Specific Demethylase 1 Inhibitors for the Treatment of Acute Myelogenous Leukemia
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 24, 页码: 22080-22103
作者:
Jiang, Hong
;
Li, Cong
;
Li, Na
;
Sheng, Li
;
Wang, Jingkai
;
Kan, Wei-Juan
;
Chen, Yuelei
;
Zhao, Dongmei
;
Guo, Dong
;
Zhou, Yu-Bo
;
Xiong, Bing
;
Li, Jia
;
Liu, Tongchao
收藏
|
浏览/下载:30/0
|
提交时间:2025/01/14
Major specialized natural products from the endangered plant
Heptacodium
miconioides,
, potential medicinal uses and insights into its longstanding unresolved systematic classification
期刊论文
PHYTOCHEMISTRY, 2024, 卷号: 228, 页码: 15
作者:
Zhao, Ze-Yu
;
Wan, Jiang
;
Chen, Hao-Wei
;
Sun, Zhong-Shuai
;
Tao, Yu-Tian
;
Tong, Yingpeng
;
Zang, Yi
;
Choo, Yeun-Mun
;
Wang, Pan
;
Li, Yue-Ling
;
Jiang, Chun-Xiao
;
Li, Junming
;
Xiong, Juan
;
Li, Jia
;
Jin, Ze-Xin
;
Hu, Jin-Feng
收藏
|
浏览/下载:37/0
|
提交时间:2024/10/21
Heptacodium miconioides
Caprifoliaceae
Systematic position
Chemotaxonomy
Enantiomeric lignans
Triterpenoids
Quinic acid derivatives
ACL inhibitory
Fortunefuroic Acid J from
Keteleeria Hainanensis
and its Dual Inhibitory Effects on ATP-Citrate Lyase and Acetyl-CoA Carboxylase
期刊论文
CHEMISTRY & BIODIVERSITY, 2024, 卷号: 21, 期号: 12, 页码: 7
作者:
Zhao, Ze-Yu
;
Zang, Yi
;
Li, Jia
;
Choo, Yeun-Mun
;
Xiong, Juan
;
Hu, Jin-Feng
收藏
|
浏览/下载:13/0
|
提交时间:2025/02/28
Keteleeria hainanensis
Pinaceae
Fortunefuroic acid
ATP-citrate lyase
Acetyl-CoA carboxylase 1
Natural products
Terpenoids
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