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Phytochemical and biological studies on rare and endangered plants endemic to China. Part XLIV. Integrated NMR/EI-MS/LC-PDA-ESIMS approach for dereplication and targeted isolation of fortunefuroic acids from Keteleeria fortunei across diverse geographical origins 期刊论文
PHYTOCHEMISTRY, 2025, 卷号: 235, 页码: 13
作者:  Zhao, Ze-Yu;  Jiang, Zhe-Lu;  Tong, Ying-Peng;  Chi, Chun-Jing;  Zang, Yi;  Choo, Yeun-Mun;  Xiong, Juan;  Li, Jia;  Hu, Jin-Feng
收藏  |  浏览/下载:25/0  |  提交时间:2025/04/24
Keteleeria fortunei  Pinaceae  Geographical origins  Integrated NMR/EI-MS/LC-PDA-ESIMS  methods  Fortunefuroic acids  ATP-Citrate lyase  
Pharmacokinetics and Safety of TPN171 (a PDE5 Inhibitor) in Patients With Mild or Moderate Hepatic Impairment Versus Participants With Normal Hepatic Function: A Phase I Study 期刊论文
CLINICAL PHARMACOLOGY IN DRUG DEVELOPMENT, 2025, 页码: 7
作者:  Zhou, Jing;  Zhang, Hong;  Ding, Yanhua;  Wang, Zhen;  Wang, Yu;  Juan, Jiaxiang;  Jiang, Zhicheng;  Chen, Hong
收藏  |  浏览/下载:1/0  |  提交时间:2025/06/23
hepatic impairment  pharmacokinetics  phosphodiesterase-5 inhibitor  TPN171  
A Phase I Study to Evaluate the Pharmacokinetics and Safety of TPN171 (a PDE5 Inhibitor) in Adults with Renal Impairment 期刊论文
CLINICAL PHARMACOLOGY IN DRUG DEVELOPMENT, 2025, 页码: 8
作者:  Fu, Ping;  Song, Yi;  Hu, Chao;  Yong, Xiaolan;  Yu, Yang;  Chen, Yi;  Wang, Ying;  Zhu, Xiaohong;  Wang, Zhen;  Wang, Yu;  Juan, Jiaxiang;  Chen, Yuan;  Miao, Jia
收藏  |  浏览/下载:2/0  |  提交时间:2025/06/23
pharmacokinetics  phosphodiesterase 5 inhibitor  renal impairment  safety  TPN171  
USP7 V517F mutation as a mechanism of inhibitor resistance 期刊论文
NATURE COMMUNICATIONS, 2025, 卷号: 16, 期号: 1, 页码: 14
作者:  Miao, Yu-Ling;  Fan, Fengying;  Cheng, Yong-Jun;  Jia, Li;  Song, Shan-Shan;  Huan, Xia-Juan;  Bao, Xu-Bin;  Ding, Jian;  Yu, Xuekui;  He, Jin-Xue
收藏  |  浏览/下载:9/0  |  提交时间:2025/05/27
New Arylalkenyl α-Pyrones from Cryptocarya densiflora 期刊论文
CHEMISTRY & BIODIVERSITY, 2025, 页码: 6
作者:  Meng, Jie;  Xue, Jun-Juan;  Miao, Lei;  Zhang, Yu;  Rao, Li;  Zhang, Chuan-Rui
收藏  |  浏览/下载:11/0  |  提交时间:2025/04/01
alpha-pyrones  Cryptocarya densiflora  cytotoxicity  quantum chemical calculations  spectroscopic data  
Benzofurans and dibenzofurans from galls on twigs of the endangered Chinese endemic tree Parrotia subaequalis and their inhibitory properties against Staphylococcus aureus and ATP-citrate lyase 期刊论文
PHYTOCHEMISTRY, 2025, 卷号: 229, 页码: 9
作者:  Zhou, Peng-Jun;  Wu, Xi-Ying;  Zhao, Ze-Yu;  Zang, Yi;  Sun, Zhong-Shuai;  Li, Yue-Ling;  Li, Na;  Xiong, Juan;  Choo, Yeun-Mun;  Jin, Ze-Xin;  Li, Jia;  Hu, Jin-Feng
收藏  |  浏览/下载:52/0  |  提交时间:2024/11/26
Parrotia subaequalis  Hamamelidaceae  Gall  Phytoalexins  Benzofuran  Dibenzofuran  Staphylococcus aureus  ATP-Citrate lyase  
π-HuB: the proteomic navigator of the human body 期刊论文
NATURE, 2024, 卷号: 636, 期号: 8042, 页码: 322-331
作者:  He, Fuchu;  Aebersold, Ruedi;  Baker, Mark S.;  Bian, Xiuwu;  Bo, Xiaochen;  Chan, Daniel W.;  Chang, Cheng;  Chen, Luonan;  Chen, Xiangmei;  Chen, Yu-Ju;  Cheng, Heping;  Collins, Ben C.;  Corrales, Fernando;  Cox, Juergen;  Weinan, E.;  Van Eyk, Jennifer E.;  Fan, Jia;  Faridi, Pouya;  Figeys, Daniel;  Gao, George Fu;  Gao, Wen;  Gao, Zu-Hua;  Goda, Keisuke;  Goh, Wilson Wen Bin;  Gu, Dongfeng;  Guo, Changjiang;  Guo, Tiannan;  He, Yuezhong;  Heck, Albert J. R.;  Hermjakob, Henning;  Hunter, Tony;  Iyer, Narayanan Gopalakrishna;  Jiang, Ying;  Jimenez, Connie R.;  Joshi, Lokesh;  Kelleher, Neil L.;  Li, Ming;  Li, Yang;  Lin, Qingsong;  Liu, Cui Hua;  Liu, Fan;  Liu, Guang-Hui;  Liu, Yansheng;  Liu, Zhihua;  Low, Teck Yew;  Lu, Ben;  Mann, Matthias;  Meng, Anming;  Moritz, Robert L.;  Nice, Edouard;  Ning, Guang;  Omenn, Gilbert S.;  Overall, Christopher M.;  Palmisano, Giuseppe;  Peng, Yaojin;  Pineau, Charles;  Poon, Terence Chuen Wai;  Purcell, Anthony W.;  Qiao, Jie;  Reddel, Roger R.;  Robinson, Phillip J.;  Roncada, Paola;  Sander, Chris;  Sha, Jiahao;  Song, Erwei;  Srivastava, Sanjeeva;  Sun, Aihua;  Sze, Siu Kwan;  Tang, Chao;  Tang, Liujun;  Tian, Ruijun;  Vizcaino, Juan Antonio;  Wang, Chanjuan;  Wang, Chen;  Wang, Xiaowen;  Wang, Xinxing;  Wang, Yan;  Weiss, Tobias;  Wilhelm, Mathias;  Winkler, Robert;  Wollscheid, Bernd;  Wong, Limsoon;  Xie, Linhai;  Xie, Wei;  Xu, Tao;  Xu, Tianhao;  Yan, Liying;  Yang, Jing;  Yang, Xiao;  Yates, John;  Yun, Tao;  Zhai, Qiwei;  Zhang, Bing;  Zhang, Hui;  Zhang, Lihua;  Zhang, Lingqiang;  Zhang, Pingwen;  Zhang, Yukui;  Zheng, Yu Zi;  Zhong, Qing;  Zhu, Yunping;  Tan, Chris Soon Heng;  Gao, Mingxia;  Gao, Qiang;  Gao, Yushun;  Guo, Xuejiang;  He, Jie;  He, Jun;  He, Qing-Yu;  Hou, Jinlin;  Huang, Canhua;  Jia, Chenxi;  Kuster, Bernhard;  Li, Chaoying;  Li, Dong;  Li, Yanchang;  Liu, Siqi;  Liu, Xiaonan;  Liu, Ya;  Liu, Zhongyang;  Lu, Haojie;  Nie, Yongzhan;  Okada, Mariko;  Qian, Guojun;  Qin, Hongqiang;  Rao, Yu;  Rao, Zihe;  Ren, Xianwen;  Ren, Yan;  Shen, Feng;  Shen, Lin;  Su, Shicheng;  Tan, Minjia;  Tang, Ben Zhong;  Tao, Sheng-Ce;  Wang, Jian;  Wang, Tong;  Wei, Liming;  Wong, Catherine C. L.;  Xie, Xiaoliang Sunney;  Xu, Li;  Xu, Ping;  Yang, Huanming;  Yang, Jianjun;  Ye, Mingliang;  Ying, Wantao;  Yu, Xiaobo;  Yuan, Yaxiang;  Zeng, Qingcun;  Zhan, Qimin;  Zhang, Xiaofei;  Zhang, Xu;  Zhang, Ying;  Zhong, Nan-Shan;  Zhou, Feng;  Zhu, Yi;  Zhang, Zemin
收藏  |  浏览/下载:16/0  |  提交时间:2025/04/01
Optimization and Biological Evaluation of Novel 1H-Pyrrolo[2,3-c]pyridin Derivatives as Potent and Reversible Lysine Specific Demethylase 1 Inhibitors for the Treatment of Acute Myelogenous Leukemia 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 24, 页码: 22080-22103
作者:  Jiang, Hong;  Li, Cong;  Li, Na;  Sheng, Li;  Wang, Jingkai;  Kan, Wei-Juan;  Chen, Yuelei;  Zhao, Dongmei;  Guo, Dong;  Zhou, Yu-Bo;  Xiong, Bing;  Li, Jia;  Liu, Tongchao
收藏  |  浏览/下载:30/0  |  提交时间:2025/01/14
Major specialized natural products from the endangered plant Heptacodium miconioides, , potential medicinal uses and insights into its longstanding unresolved systematic classification 期刊论文
PHYTOCHEMISTRY, 2024, 卷号: 228, 页码: 15
作者:  Zhao, Ze-Yu;  Wan, Jiang;  Chen, Hao-Wei;  Sun, Zhong-Shuai;  Tao, Yu-Tian;  Tong, Yingpeng;  Zang, Yi;  Choo, Yeun-Mun;  Wang, Pan;  Li, Yue-Ling;  Jiang, Chun-Xiao;  Li, Junming;  Xiong, Juan;  Li, Jia;  Jin, Ze-Xin;  Hu, Jin-Feng
收藏  |  浏览/下载:37/0  |  提交时间:2024/10/21
Heptacodium miconioides  Caprifoliaceae  Systematic position  Chemotaxonomy  Enantiomeric lignans  Triterpenoids  Quinic acid derivatives  ACL inhibitory  
Fortunefuroic Acid J from Keteleeria Hainanensis and its Dual Inhibitory Effects on ATP-Citrate Lyase and Acetyl-CoA Carboxylase 期刊论文
CHEMISTRY & BIODIVERSITY, 2024, 卷号: 21, 期号: 12, 页码: 7
作者:  Zhao, Ze-Yu;  Zang, Yi;  Li, Jia;  Choo, Yeun-Mun;  Xiong, Juan;  Hu, Jin-Feng
收藏  |  浏览/下载:13/0  |  提交时间:2025/02/28
Keteleeria hainanensis  Pinaceae  Fortunefuroic acid  ATP-citrate lyase  Acetyl-CoA carboxylase 1  Natural products  Terpenoids  
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