KMS@SIMM

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Development of novel epoxyketone macrocyclic peptidyl proteasome inhibitors through OPA-mediated one-step cyclization of unprotected peptides 期刊论文
BIOORGANIC CHEMISTRY, 2025, 卷号: 156, 页码: 16
作者:  Zeng, Gongruixue;  Xu, Gaoya;  Gao, Lixin;  Zheng, Xiaoli;  Chi, Xinglong;  Shen, Zheyuan;  Cao, Yu;  Xi, Jianjun;  Che, Jinxin;  Dong, Xiaowu;  Shi, Yaoli;  Ma, Jiayi;  Zhang, Chong;  Zeng, Linghui;  Zhu, Huajian;  Shao, Jiaan;  Zhou, Yubo;  Li, Jia;  Zhang, Jiankang
收藏  |  浏览/下载:15/0  |  提交时间:2025/04/01
Proteasome inhibitors  Macrocycle  Stability  Anti-cancer activities  
Discovery of a potential hematologic malignancies therapy: Selective and potent HDAC7 PROTAC degrader targeting non-enzymatic function 期刊论文
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 3, 页码: 1659-1679
作者:  Jin, Yuheng;  Qi, Xuxin;  Yu, Xiaoli;  Cheng, Xirui;  Chen, Boya;  Wu, Mingfei;  Zhang, Jingyu;  Yin, Hao;  Lu, Yang;  Zhou, Yihui;  Pang, Ao;  Lin, Yushen;  Jiang, Li;  Shi, Qiuqiu;  Geng, Shuangshuang;  Zhou, Yubo;  Yao, Xiaojun;  Li, Linjie;  Duan, Haiting;  Che, Jinxin;  Cao, Ji;  He, Qiaojun;  Dong, Xiaowu
收藏  |  浏览/下载:1/0  |  提交时间:2025/06/23
HDAC7  PROTAC  Selectivity  Hematologic malignancies  Non-enzymatic function  
The critical role of MLKL in hemorrhagic stroke and the therapeutic potential of its associated protein network 期刊论文
FRONTIERS IN CELL AND DEVELOPMENTAL BIOLOGY, 2025, 卷号: 12, 页码: 12
作者:  Wang, Yi;  Xu, Moran;  Zuo, Xiaoli;  Wang, Sheng;  Yu, Yong;  Gao, Zhaobing;  Qie, Jingbo;  Jiang, Ye;  Huang, Fang;  Xia, Bingqing
收藏  |  浏览/下载:21/0  |  提交时间:2025/04/01
mlkl  ICH  hemorrhagic stroke  neuroinflammation  LC-MS/MS  
Auto-RapTAC: A Versatile and Sustainable Platform for the Automated Rapid Synthesis and Evaluation of PROTAC 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 15
作者:  Chen, Jiexuan;  Wu, Mingfei;  Mo, Jun;  Hong, Ju;  Wang, Wei;  Jin, Yuheng;  Mao, Xinfei;  Liao, Xueyan;  Li, Kailin;  Yu, Xiaoli;  Chen, Sikang;  Zeng, Shenxin;  Huang, Wenhai;  Xu, Hongxia;  Wu, Jian;  Cao, Ji;  Zhou, Yubo;  Ying, Meidan;  Zhu, Chengliang;  He, Qiaojun;  Zhang, Bo;  Lin, Nengming;  Dong, Xiaowu;  Che, Jinxin
收藏  |  浏览/下载:20/0  |  提交时间:2025/04/01
Sevoflurane Alters Serum Metabolites in Elders and Aging Mice and Increases Inflammation in Hippocampus 期刊论文
JOURNAL OF INFLAMMATION RESEARCH, 2024, 卷号: 17, 页码: 1241-1253
作者:  Wang, Tingting;  Wu, Xia;  Zhao, Xiaoli;  Li, Jiaqi;  Yu, Jian;  Sheng, Maozheng;  Gao, Mingyuan;  Cao, Yutang;  Wang, Jiawen;  Guo, Xiaozhen;  Zeng, Kai
收藏  |  浏览/下载:42/0  |  提交时间:2024/04/09
sevoflurane  hippocampus  neuroinflammation  RNA-seq  metabolomics  isatin  
Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 18
作者:  Zhang, Jingyu;  Duan, Haiting;  Gui, Renzhao;  Wu, Mingfei;  Shen, Liteng;  Jin, Yuheng;  Pang, Ao;  Yu, Xiaoli;  Zeng, Shenxin;  Zhang, Bo;  Lin, Nengming;  Huang, Wenhai;  Wang, Yuwei;  Yao, Xiaojun;  Li, Jia;  Dong, Xiaowu;  Zhou, Yubo;  Che, Jinxin
收藏  |  浏览/下载:77/0  |  提交时间:2023/12/19
Acute myeloid leukemia  Bromodomain-containing protein 9  Proteolysis-targeting chimera  Orally bioavailable  Docking  
SARS-CoV-2 envelope protein causes acute respiratory distress syndrome (ARDS)-like pathological damages and constitutes an antiviral target 期刊论文
CELL RESEARCH, 2021, 页码: 14
作者:  Xia, Bingqing;  Shen, Xurui;  He, Yang;  Pan, Xiaoyan;  Liu, Feng-Liang;  Wang, Yi;  Yang, Feipu;  Fang, Sui;  Wu, Yan;  Duan, Zilei;  Zuo, Xiaoli;  Xie, Zhuqing;  Jiang, Xiangrui;  Xu, Ling;  Chi, Hao;  Li, Shuangqu;  Meng, Qian;  Zhou, Hu;  Zhou, Yubo;  Cheng, Xi;  Xin, Xiaoming;  Jin, Lin;  Zhang, Hai-Lin;  Yu, Dan-Dan;  Li, Ming-Hua;  Feng, Xiao-Li;  Chen, Jiekai;  Jiang, Hualiang;  Xiao, Gengfu;  Zheng, Yong-Tang;  Zhang, Lei-Ke;  Shen, Jingshan;  Li, Jia;  Gao, Zhaobing
收藏  |  浏览/下载:96/0  |  提交时间:2021/08/17
Interfering MSN-NONO complex-activated CREB signaling serves as a therapeutic strategy for triple-negative breast cancer 期刊论文
SCIENCE ADVANCES, 2020, 卷号: 6, 期号: 8, 页码: 13
作者:  Qin, Yuanyuan;  Chen, Weilong;  Jiang, Guojuan;  Zhou, Lei;  Yang, Xiaoli;  Li, Hongqi;  He, Xueyan;  Wang, Han-lin;  Zhou, Yu-bo;  Huang, Shenglin;  Liu, Suling
收藏  |  浏览/下载:70/0  |  提交时间:2020/07/01
Pharmacokinetics-Driven Optimization of 4(3H)-Pyrimidinones as Phosphodiesterase Type 5 Inhibitors Leading to TPN171, a Clinical Candidate for the Treatment of Pulmonary Arterial Hypertension 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 10, 页码: 4979-4990
作者:  Wang, Zhen;  Jiang, Xiangrui;  Zhang, Xianglei;  Tian, Guanghui;  Yang, Rulei;  Wu, Jianzhong;  Zou, Xiaoli;  Liu, Zheng;  Yang, Xiaojun;  Wu, Chunhui;  Shi, Jing;  Li, Jianfeng;  Suo, Jin;  Wang, Yu;  Zhang, Rongxia;  Xu, Zhijian;  Gong, Xudong;  He, Yang;  Zhu, Weiliang;  Aisa, Haji Akber;  Jiang, Hualiang;  Xu, Yechun;  Shen, Jingshan
收藏  |  浏览/下载:72/0  |  提交时间:2020/07/01
A G3BP1-Interacting lncRNA Promotes Ferroptosis and Apoptosis in Cancer via Nuclear Sequestration of p53 期刊论文
CANCER RESEARCH, 2018, 卷号: 78, 期号: 13, 页码: 3484-3496
作者:  Mao, Chao;  Wang, Xiang;  Liu, Yating;  Wang, Min;  Bin Yan;  Jiang, Yiqun;  Shi, Ying;  Shen, Yi;  Liu, Xiaoli;  Lai, Weiwei;  Yang, Rui;  Xiao, Desheng;  Cheng, Yan;  Liu, Shuang;  Zhou, Hu;  Cao, Ya;  Yu, Weishi;  Muegge, Kathrin;  Yu, Herbert;  Tao, Yongguang
收藏  |  浏览/下载:87/0  |  提交时间:2019/01/08
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