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中国科学院上海药物研究所机构知识库
Knowledge Management System of Shanghai Institute of Materia Medica, CAS
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Development of novel epoxyketone macrocyclic peptidyl proteasome inhibitors through OPA-mediated one-step cyclization of unprotected peptides
期刊论文
BIOORGANIC CHEMISTRY, 2025, 卷号: 156, 页码: 16
作者:
Zeng, Gongruixue
;
Xu, Gaoya
;
Gao, Lixin
;
Zheng, Xiaoli
;
Chi, Xinglong
;
Shen, Zheyuan
;
Cao, Yu
;
Xi, Jianjun
;
Che, Jinxin
;
Dong, Xiaowu
;
Shi, Yaoli
;
Ma, Jiayi
;
Zhang, Chong
;
Zeng, Linghui
;
Zhu, Huajian
;
Shao, Jiaan
;
Zhou, Yubo
;
Li, Jia
;
Zhang, Jiankang
收藏
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浏览/下载:15/0
|
提交时间:2025/04/01
Proteasome inhibitors
Macrocycle
Stability
Anti-cancer activities
Discovery of a potential hematologic malignancies therapy: Selective and potent HDAC7 PROTAC degrader targeting non-enzymatic function
期刊论文
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 3, 页码: 1659-1679
作者:
Jin, Yuheng
;
Qi, Xuxin
;
Yu, Xiaoli
;
Cheng, Xirui
;
Chen, Boya
;
Wu, Mingfei
;
Zhang, Jingyu
;
Yin, Hao
;
Lu, Yang
;
Zhou, Yihui
;
Pang, Ao
;
Lin, Yushen
;
Jiang, Li
;
Shi, Qiuqiu
;
Geng, Shuangshuang
;
Zhou, Yubo
;
Yao, Xiaojun
;
Li, Linjie
;
Duan, Haiting
;
Che, Jinxin
;
Cao, Ji
;
He, Qiaojun
;
Dong, Xiaowu
收藏
|
浏览/下载:1/0
|
提交时间:2025/06/23
HDAC7
PROTAC
Selectivity
Hematologic malignancies
Non-enzymatic function
The critical role of MLKL in hemorrhagic stroke and the therapeutic potential of its associated protein network
期刊论文
FRONTIERS IN CELL AND DEVELOPMENTAL BIOLOGY, 2025, 卷号: 12, 页码: 12
作者:
Wang, Yi
;
Xu, Moran
;
Zuo, Xiaoli
;
Wang, Sheng
;
Yu, Yong
;
Gao, Zhaobing
;
Qie, Jingbo
;
Jiang, Ye
;
Huang, Fang
;
Xia, Bingqing
收藏
|
浏览/下载:21/0
|
提交时间:2025/04/01
mlkl
ICH
hemorrhagic stroke
neuroinflammation
LC-MS/MS
Auto-RapTAC: A Versatile and Sustainable Platform for the Automated Rapid Synthesis and Evaluation of PROTAC
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 15
作者:
Chen, Jiexuan
;
Wu, Mingfei
;
Mo, Jun
;
Hong, Ju
;
Wang, Wei
;
Jin, Yuheng
;
Mao, Xinfei
;
Liao, Xueyan
;
Li, Kailin
;
Yu, Xiaoli
;
Chen, Sikang
;
Zeng, Shenxin
;
Huang, Wenhai
;
Xu, Hongxia
;
Wu, Jian
;
Cao, Ji
;
Zhou, Yubo
;
Ying, Meidan
;
Zhu, Chengliang
;
He, Qiaojun
;
Zhang, Bo
;
Lin, Nengming
;
Dong, Xiaowu
;
Che, Jinxin
收藏
|
浏览/下载:20/0
|
提交时间:2025/04/01
Sevoflurane Alters Serum Metabolites in Elders and Aging Mice and Increases Inflammation in Hippocampus
期刊论文
JOURNAL OF INFLAMMATION RESEARCH, 2024, 卷号: 17, 页码: 1241-1253
作者:
Wang, Tingting
;
Wu, Xia
;
Zhao, Xiaoli
;
Li, Jiaqi
;
Yu, Jian
;
Sheng, Maozheng
;
Gao, Mingyuan
;
Cao, Yutang
;
Wang, Jiawen
;
Guo, Xiaozhen
;
Zeng, Kai
收藏
|
浏览/下载:42/0
|
提交时间:2024/04/09
sevoflurane
hippocampus
neuroinflammation
RNA-seq
metabolomics
isatin
Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 18
作者:
Zhang, Jingyu
;
Duan, Haiting
;
Gui, Renzhao
;
Wu, Mingfei
;
Shen, Liteng
;
Jin, Yuheng
;
Pang, Ao
;
Yu, Xiaoli
;
Zeng, Shenxin
;
Zhang, Bo
;
Lin, Nengming
;
Huang, Wenhai
;
Wang, Yuwei
;
Yao, Xiaojun
;
Li, Jia
;
Dong, Xiaowu
;
Zhou, Yubo
;
Che, Jinxin
收藏
|
浏览/下载:77/0
|
提交时间:2023/12/19
Acute myeloid leukemia
Bromodomain-containing protein 9
Proteolysis-targeting chimera
Orally bioavailable
Docking
SARS-CoV-2 envelope protein causes acute respiratory distress syndrome (ARDS)-like pathological damages and constitutes an antiviral target
期刊论文
CELL RESEARCH, 2021, 页码: 14
作者:
Xia, Bingqing
;
Shen, Xurui
;
He, Yang
;
Pan, Xiaoyan
;
Liu, Feng-Liang
;
Wang, Yi
;
Yang, Feipu
;
Fang, Sui
;
Wu, Yan
;
Duan, Zilei
;
Zuo, Xiaoli
;
Xie, Zhuqing
;
Jiang, Xiangrui
;
Xu, Ling
;
Chi, Hao
;
Li, Shuangqu
;
Meng, Qian
;
Zhou, Hu
;
Zhou, Yubo
;
Cheng, Xi
;
Xin, Xiaoming
;
Jin, Lin
;
Zhang, Hai-Lin
;
Yu, Dan-Dan
;
Li, Ming-Hua
;
Feng, Xiao-Li
;
Chen, Jiekai
;
Jiang, Hualiang
;
Xiao, Gengfu
;
Zheng, Yong-Tang
;
Zhang, Lei-Ke
;
Shen, Jingshan
;
Li, Jia
;
Gao, Zhaobing
收藏
|
浏览/下载:96/0
|
提交时间:2021/08/17
Interfering MSN-NONO complex-activated CREB signaling serves as a therapeutic strategy for triple-negative breast cancer
期刊论文
SCIENCE ADVANCES, 2020, 卷号: 6, 期号: 8, 页码: 13
作者:
Qin, Yuanyuan
;
Chen, Weilong
;
Jiang, Guojuan
;
Zhou, Lei
;
Yang, Xiaoli
;
Li, Hongqi
;
He, Xueyan
;
Wang, Han-lin
;
Zhou, Yu-bo
;
Huang, Shenglin
;
Liu, Suling
收藏
|
浏览/下载:70/0
|
提交时间:2020/07/01
Pharmacokinetics-Driven Optimization of 4(3H)-Pyrimidinones as Phosphodiesterase Type 5 Inhibitors Leading to TPN171, a Clinical Candidate for the Treatment of Pulmonary Arterial Hypertension
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 10, 页码: 4979-4990
作者:
Wang, Zhen
;
Jiang, Xiangrui
;
Zhang, Xianglei
;
Tian, Guanghui
;
Yang, Rulei
;
Wu, Jianzhong
;
Zou, Xiaoli
;
Liu, Zheng
;
Yang, Xiaojun
;
Wu, Chunhui
;
Shi, Jing
;
Li, Jianfeng
;
Suo, Jin
;
Wang, Yu
;
Zhang, Rongxia
;
Xu, Zhijian
;
Gong, Xudong
;
He, Yang
;
Zhu, Weiliang
;
Aisa, Haji Akber
;
Jiang, Hualiang
;
Xu, Yechun
;
Shen, Jingshan
收藏
|
浏览/下载:72/0
|
提交时间:2020/07/01
A G3BP1-Interacting lncRNA Promotes Ferroptosis and Apoptosis in Cancer via Nuclear Sequestration of p53
期刊论文
CANCER RESEARCH, 2018, 卷号: 78, 期号: 13, 页码: 3484-3496
作者:
Mao, Chao
;
Wang, Xiang
;
Liu, Yating
;
Wang, Min
;
Bin Yan
;
Jiang, Yiqun
;
Shi, Ying
;
Shen, Yi
;
Liu, Xiaoli
;
Lai, Weiwei
;
Yang, Rui
;
Xiao, Desheng
;
Cheng, Yan
;
Liu, Shuang
;
Zhou, Hu
;
Cao, Ya
;
Yu, Weishi
;
Muegge, Kathrin
;
Yu, Herbert
;
Tao, Yongguang
收藏
|
浏览/下载:87/0
|
提交时间:2019/01/08
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