KMS@SIMM

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Screening and preparation of nanobodies for SIGLEC-15 detection 期刊论文
PROTEIN EXPRESSION AND PURIFICATION, 2025, 卷号: 229, 页码: 9
作者:  Zhao, Shuaiying;  Li, Lingyun;  Lan, Zhongyun;  Hou, Xiangyun;  Huang, Ruimin;  Jin, Quanfang;  Huang, Qiting;  Jia, Li;  Kong, Yingying;  Wen, Jianchuan;  Qiao, Huarui;  Wang, Yiang;  Xu, Yiwen;  Zhang, Dongna;  Geng, Yong;  Xu, Jianfeng;  Dai, Yuanyuan
收藏  |  浏览/下载:82/0  |  提交时间:2025/04/01
SIGLEC-15  Nanobody  Expression  Purification  
Novel Aryl Sulfonium Modification on Vancomycin to Tackle MRSA and VRE In Vitro and In Vivo through Dual Enhanced Cell-Wall and Membrane Inhibition 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 8, 页码: 8310-8329
作者:  Xie, Yuanyuan;  Wang, Xiaowen;  Chang, Taopeng;  Chen, Zhifu;  Luo, Youhong;  Zhang, Jingwen;  Wang, Hui;  Dong, Jinhua;  Chen, Feifei;  Zhang, Jinyong;  Guan, Dongliang
收藏  |  浏览/下载:2/0  |  提交时间:2025/06/23
A Rationally Designed Sulfonium Lipoglycopeptide with Micelles Self-Assembly to Combat Multidrug Resistance via Dual Enhanced Cell Wall-Membrane Inhibition and T7SS Proteins Downregulation 期刊论文
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2025, 卷号: 147, 期号: 15, 页码: 12587-12603
作者:  Xie, Yuanyuan;  Wang, Xiaowen;  Li, Fang;  Chen, Zhifu;  Li, Qun;  Liu, Shuhui;  Zhang, Jingwen;  Wang, Hui;  Wu, Zhenyong;  Zhang, Jinyong;  Guan, Dongliang
收藏  |  浏览/下载:5/0  |  提交时间:2025/05/27
Revolutionizing fixed-dose combinations with long-acting microsphere 期刊论文
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2025, 卷号: 207, 页码: 12
作者:  Hu, Zhenhua;  Xiao, Xiao;  Zhang, Guiyun;  Li, Yuanyuan
收藏  |  浏览/下载:88/0  |  提交时间:2025/04/01
Fixed-dose combinations  Microsphere  Chronic disease  Long-acting  
Deep Learning Enhanced Near Infrared-II Imaging and Image-Guided Small Interfering Ribonucleic Acid Therapy of Ischemic Stroke 期刊论文
ACS NANO, 2025, 卷号: 19, 期号: 10, 页码: 10323-10336
作者:  Yu, Kai;  Fu, Lidan;  Chao, Yu;  Zeng, Xiaodong;  Zhang, Yonggang;  Chen, Yuanyuan;  Gao, Jialu;  Lu, Binchun;  Zhu, Hua;  Gu, Lijuan;  Xiong, Xiaoxing;  Hu, Zhenhua;  Hong, Xuechuan;  Xiao, Yuling
收藏  |  浏览/下载:11/0  |  提交时间:2025/04/24
ischemic stroke  small interferingRNA therapy  near-infrared II imaging  blood-brainbarrier  deep learning  
Near-Infrared Activatable Copper Nanoplatforms Synergize with the 5-Azacytidine Prodrug to Potentiate Cuproptosis 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2024, 页码: 13
作者:  Wang, Shuo;  Liu, Yishen;  Su, Mengya;  Wang, Yuanyuan;  Wang, Wenda;  Wang, Wuyin;  Yang, Qichao;  Zhang, Zhiyun;  Hong, Xuechuan;  Sun, Zhijun;  Xiao, Yuling
收藏  |  浏览/下载:43/0  |  提交时间:2024/12/16
cuproptosis  near-infrared light  photocatalysis  antitumor therapy  ferredoxin 1  
Prediction of Multi-Pharmacokinetics Property in Multi-Species: Bayesian Neural Network Stacking Model with Uncertainty 期刊论文
MOLECULAR PHARMACEUTICS, 2024, 页码: 16
作者:  Zhang, Yuanyuan;  Xie, Zhiyin;  Xiao, Fu;  Yu, Jie;  Fan, Zhehuan;  Sun, Shihui;  Shi, Jiangshan;  Fu, Zunyun;  Li, Xutong;  Wang, Dingyan;  Zheng, Mingyue;  Luo, Xiaomin
收藏  |  浏览/下载:35/0  |  提交时间:2024/12/11
pharmacokinetic parameters  machine learning  uncertainty  stacking  multitask learning  ADME  
Single Amine or Guanidine Modification on Norvancomycin and Vancomycin to Overcome Multidrug-Resistance through Augmented Lipid II Binding and Increased Membrane Activity 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 22, 页码: 20639-20663
作者:  Bian, Xiaolei;  Chen, Zhifu;  Li, Fang;  Xie, Yuanyuan;  Li, Yi;  Luo, Youhong;  Zou, Xiangman;  Wang, Hui;  Zhang, Jingwen;  Wang, Xiaowen;  Zhang, Jinyong;  Guan, Dongliang
收藏  |  浏览/下载:22/0  |  提交时间:2024/12/11
Discovery of pyridazinone derivatives bearing tetrahydroimidazo[1,2- a ] pyrazine scaffold as potent inhibitors of transient receptor potential canonical 5 to ameliorate hypertension-induced renal injury in rats 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 275, 页码: 18
作者:  Xu, Yuanyuan;  Ren, Younan;  Zhang, Jie;  Niu, Bo;  Liu, Mengru;  Xu, Tifei;  Zhang, Xian;  Shen, Jianhua;  Wang, Kai;  Cao, Zhengyu
收藏  |  浏览/下载:301/0  |  提交时间:2024/08/22
Pyridazinone  Tetrahydroimidazo[1,2-a]pyrazine  Transient receptor potential canonical 5  Chronic kidney disease  Focal segmental glomerulosclerosis  
De novo design of SARS-CoV-2 main protease inhibitors with characteristic binding modes 期刊论文
STRUCTURE, 2024, 卷号: 32, 期号: 9, 页码: 12
作者:  Zhu, Yan;  Meng, Jiaolong;  Feng, Bo;  Zhao, Yao;  Zang, Yi;  Lu, Lingling;  Su, Mingbo;  Yang, Qi;  Zhang, Qi;  Feng, Lu;  Zhao, Jinyi;  Shao, Maolin;  Ma, Yuanyuan;  Yang, Xiuna;  Yang, Haitao;  Li, Jia;  Jiang, Xuefeng;  Rao, Zihe
收藏  |  浏览/下载:35/0  |  提交时间:2024/10/21
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