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Pharmacokinetics, mass balance, and metabolism of [14C]PLB1004, a selective and irreversible EGFR-TKI in humans 期刊论文
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2025, 卷号: 95, 期号: 1, 页码: 14
作者:  Liu, Donghui;  Li, Qian;  Yan, Shu;  Zhang, Xinyue;  Li, Weiqiang;  Wang, Feiyu;  Gao, Lei;  Geng, Fei;  Zhou, Haiyan;  Ye, Panpan;  Zhao, Furong;  Xue, Weizhe;  Zhang, Peilong;  Diao, Xingxing;  Zhao, Wei
收藏  |  浏览/下载:39/0  |  提交时间:2025/04/01
PLB1004  [C-14]PLB1004  Radioactivity  Mass balance  EGFR-TKI  
BMAL1/PGC1a4-FNDC5/irisin axis impacts distinct outcomes of time-of-day resistance exercise 期刊论文
JOURNAL OF SPORT AND HEALTH SCIENCE, 2025, 卷号: 14, 页码: 23
作者:  Guo, Mingwei;  Shen, Fei;  Guo, Xiaozhen;  Zhang, Jun;  Ma, Ying;  Wu, Xia;  Zuo, Hui;  Yao, Jing;  Hu, Yepeng;  Wang, Dongmei;  Li, Yu;  Li, Jin;  Qiu, Jin;  Yu, Jian;  Meng, Meiyao;  Zheng, Ying;  Chen, Xin;  Gong, Mingkai;  Liu, Kailin;  Jin, Ling;  Ren, Xiangyu;  Zhang, Qiang;  Zhao, Yu;  Gu, Xuejiang;  Shen, Feixia;  Li, Dali;  Gao, Liangcai;  Liu, Chang;  Zhou, Fei;  Li, Mian;  Wang, Jiqiu;  Ding, Shuzhe;  Ma, Xinran;  Lu, Jian;  Xie, Cen;  Xiao, Junjie;  Xu, Lingyan
收藏  |  浏览/下载:51/0  |  提交时间:2025/04/01
Daily variance  Circadian  Muscle strength  Metabolic benefits  Resistance exercise  
Phytochemical and biological studies on rare and endangered plants endemic to China. Part XLIV. Integrated NMR/EI-MS/LC-PDA-ESIMS approach for dereplication and targeted isolation of fortunefuroic acids from Keteleeria fortunei across diverse geographical origins 期刊论文
PHYTOCHEMISTRY, 2025, 卷号: 235, 页码: 13
作者:  Zhao, Ze-Yu;  Jiang, Zhe-Lu;  Tong, Ying-Peng;  Chi, Chun-Jing;  Zang, Yi;  Choo, Yeun-Mun;  Xiong, Juan;  Li, Jia;  Hu, Jin-Feng
收藏  |  浏览/下载:30/0  |  提交时间:2025/04/24
Keteleeria fortunei  Pinaceae  Geographical origins  Integrated NMR/EI-MS/LC-PDA-ESIMS  methods  Fortunefuroic acids  ATP-Citrate lyase  
Screening and functional characterization of nanobodies targeting the transferrin receptor 期刊论文
PROTEIN EXPRESSION AND PURIFICATION, 2025, 卷号: 231, 页码: 7
作者:  Ding, Yuting;  Jia, Li;  Geng, Qifubo;  Liu, Yan;  Guo, Shaojue;  Zhao, Shuaiying;  Kong, Yingying;  Jin, Quanfang;  Xu, Guangxu;  Xu, Jianfeng
收藏  |  浏览/下载:26/0  |  提交时间:2025/05/27
Transferrin receptor (TfR1)  Nanobody screening  Cancer therapy  
(+)-Borneol Enhances the Antiseizure Effects of Retigabine by both Pharmacokinetic and Pharmacodynamic Interaction 期刊论文
NEUROCHEMICAL RESEARCH, 2025, 卷号: 50, 期号: 3, 页码: 13
作者:  Xu, Haiyan;  Wu, Zhidan;  Wang, Pei;  Gong, Jili;  Qiu, Li;  Gu, Yueling;  Zhan, Li;  Tian, Fuyun;  Gao, Zhaobing
收藏  |  浏览/下载:9/0  |  提交时间:2025/06/23
Epilepsy  Retigabine  (+)-Borneol  Synergistic interaction  KCNQ channels  
Targeted degradation of GOLM1 by CC-885 via CRL4-CRBN E3 ligase inhibits hepatocellular carcinoma progression 期刊论文
CELLULAR SIGNALLING, 2025, 卷号: 130, 页码: 15
作者:  He, Jingliang;  Guo, Jingli;  Liu, Shunfang;  Li, Hanxue;  Ma, Yuanyuan;  Ma, Shaojie;  Hu, Zhongke;  Zhao, Wensi;  Tan, Minjia;  Liu, Wei;  Liu, Bin
收藏  |  浏览/下载:20/0  |  提交时间:2025/04/24
Hepatocellular carcinoma  CC-885  GOLM1  Ubiquitination  Apoptosis  CRBN  
Dehydrotrametenolic acid methyl ester, a triterpenoid of Poria cocos, alleviates non-alcoholic steatohepatitis by suppressing NLRP3 inflammasome activation via targeting Caspase-1 in mice 期刊论文
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 17
作者:  Xia, Ling-yan;  Yu, Nai-rong;  Huang, Su-ling;  Qu, Hui;  Qin, Li;  Zhao, Qin-shi;  Leng, Ying
收藏  |  浏览/下载:7/0  |  提交时间:2025/06/23
non-alcoholic steatohepatitis  dehydrotrametenolic acid methyl ester  NLRP3 inflammasome  caspase-1  macrophage-hepatocyte/HSC crosstalk  
Screening and preparation of nanobodies for SIGLEC-15 detection 期刊论文
PROTEIN EXPRESSION AND PURIFICATION, 2025, 卷号: 229, 页码: 9
作者:  Zhao, Shuaiying;  Li, Lingyun;  Lan, Zhongyun;  Hou, Xiangyun;  Huang, Ruimin;  Jin, Quanfang;  Huang, Qiting;  Jia, Li;  Kong, Yingying;  Wen, Jianchuan;  Qiao, Huarui;  Wang, Yiang;  Xu, Yiwen;  Zhang, Dongna;  Geng, Yong;  Xu, Jianfeng;  Dai, Yuanyuan
收藏  |  浏览/下载:88/0  |  提交时间:2025/04/01
SIGLEC-15  Nanobody  Expression  Purification  
"Targeting AhR suppresses hepatocyte ferroptosis in MASH by regulating the Pten/Akt/β catenin axis" [Biochem. Pharmacol. 232 (2025) 116711] 期刊论文
BIOCHEMICAL PHARMACOLOGY, 2025, 卷号: 235, 页码: 1
作者:  Ma, Chenhui;  Han, Li;  Zhao, Wenxuan;  Chen, Feihong;  Huang, Ruimin;  Pang, Cheng Heng;  Zhu, Zheying;  Pan, Guoyu
收藏  |  浏览/下载:13/0  |  提交时间:2025/04/24
Neuronal CCL2 responds to hyperglycaemia and contributes to anxiety disorders in the context of diabetes 期刊论文
NATURE METABOLISM, 2025, 卷号: 7, 期号: 5, 页码: 39
作者:  Pan, Kaijun;  Gao, Yanan;  Zong, Haichao;  Zhang, Yongmei;  Qi, Yingbei;  Wang, Hanlin;  Chen, Wengang;  Zhou, Ting;  Zhao, Jinwen;  Yin, Tao;  Guo, Haoran;  Wang, Min;  Wang, Hanmin;  Pang, Tao;  Zang, Yi;  Li, Jia
收藏  |  浏览/下载:22/0  |  提交时间:2025/06/23
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